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Bioorg Med Chem Lett
; 20(11): 3219-22, 2010 Jun 01.
Article
de Anglais
| MEDLINE
| ID: mdl-20457517
RÉSUMÉ
Elaboration of our previously disclosed spiropiperidine template led to the development of a series of novel CCR5 antagonists. Results of SAR exploration and preliminary lead characterization are described.