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9H-Xanthene-9-carboxylic acid [1,2,4]oxadiazol-3-yl- and (2H-tetrazol-5-yl)-amides as potent, orally available mGlu1 receptor enhancers.
Vieira, Eric; Huwyler, Jörg; Jolidon, Synèse; Knoflach, Frédéric; Mutel, Vincent; Wichmann, Jürgen.
Affiliation
  • Vieira E; Pharma Division, Discovery Research, F. Hoffmann-La Roche Ltd., CH-4070 Basel, Switzerland. eric.vieira@roche.com
Bioorg Med Chem Lett ; 15(20): 4628-31, 2005 Oct 15.
Article in En | MEDLINE | ID: mdl-16099654
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Collection: 01-internacional Database: MEDLINE Main subject: Oxadiazoles / Tetrazoles / Receptors, Metabotropic Glutamate / Excitatory Amino Acid Agonists Limits: Animals Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2005 Document type: Article Affiliation country:
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Collection: 01-internacional Database: MEDLINE Main subject: Oxadiazoles / Tetrazoles / Receptors, Metabotropic Glutamate / Excitatory Amino Acid Agonists Limits: Animals Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2005 Document type: Article Affiliation country: