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Rational design, synthesis, and structure-activity relationship of benzoxazolones: new potent mglu5 receptor antagonists based on the fenobam structure.
Ceccarelli, Simona M; Jaeschke, Georg; Buettelmann, Bernd; Huwyler, Jörg; Kolczewski, Sabine; Peters, Jens-Uwe; Prinssen, Eric; Porter, Richard; Spooren, Will; Vieira, Eric.
Affiliation
  • Ceccarelli SM; Pharmaceutical Division, Discovery Research, F. Hoffmann-La Roche Ltd,CH-4070 Basel, Switzerland. Simona_m.ceccarelli@roche.com
Bioorg Med Chem Lett ; 17(5): 1302-6, 2007 Mar 01.
Article in En | MEDLINE | ID: mdl-17189691
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Collection: 01-internacional Database: MEDLINE Main subject: Anti-Anxiety Agents / Benzoxazoles / Receptors, Metabotropic Glutamate Limits: Animals Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2007 Document type: Article Affiliation country:
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Collection: 01-internacional Database: MEDLINE Main subject: Anti-Anxiety Agents / Benzoxazoles / Receptors, Metabotropic Glutamate Limits: Animals Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2007 Document type: Article Affiliation country: