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Synthesis and characterization of 8-ethynyl-1,3-dihydro-benzo[b][1,4]diazepin-2-one derivatives: new potent non-competitive metabotropic glutamate receptor 2/3 antagonists. Part 1.
Woltering, Thomas J; Adam, Geo; Alanine, Alexander; Wichmann, Jürgen; Knoflach, Frédéric; Mutel, Vincent; Gatti, Silvia.
Affiliation
  • Woltering TJ; F. Hoffmann-La Roche Ltd, Pharma Discovery Chemistry, CNS CH-4070 Basel, Switzerland.
Bioorg Med Chem Lett ; 17(24): 6811-5, 2007 Dec 15.
Article in En | MEDLINE | ID: mdl-17964783
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Collection: 01-internacional Database: MEDLINE Main subject: Azepines / Receptors, Metabotropic Glutamate Limits: Animals Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2007 Document type: Article Affiliation country:
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Collection: 01-internacional Database: MEDLINE Main subject: Azepines / Receptors, Metabotropic Glutamate Limits: Animals Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2007 Document type: Article Affiliation country: