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Structural modifications of N-arylamide oxadiazoles: Identification of N-arylpiperidine oxadiazoles as potent and selective agonists of CB2.
DiMauro, Erin F; Buchanan, John L; Cheng, Alan; Emkey, Renee; Hitchcock, Stephen A; Huang, Liyue; Huang, Ming Y; Janosky, Brett; Lee, Josie H; Li, Xingwen; Martin, Matthew W; Tomlinson, Susan A; White, Ryan D; Zheng, Xiao Mei; Patel, Vinod F; Fremeau, Robert T.
Affiliation
  • DiMauro EF; Department of Medicinal Chemistry, Amgen Inc., One Kendall Square, Building 1000, Cambridge, MA 02139, USA. edimauro@amgen.com
Bioorg Med Chem Lett ; 18(15): 4267-74, 2008 Aug 01.
Article in En | MEDLINE | ID: mdl-18640038

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Oxadiazoles / Microsomes, Liver / Receptor, Cannabinoid, CB2 Type of study: Diagnostic_studies Limits: Animals / Humans Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2008 Document type: Article Affiliation country: Country of publication:

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Oxadiazoles / Microsomes, Liver / Receptor, Cannabinoid, CB2 Type of study: Diagnostic_studies Limits: Animals / Humans Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2008 Document type: Article Affiliation country: Country of publication: