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Discovery of the First Potent and Selective Inhibitor of Centromere-Associated Protein E: GSK923295.
Qian, Xiangping; McDonald, Andrew; Zhou, Han-Jie; Adams, Nicholas D; Parrish, Cynthia A; Duffy, Kevin J; Fitch, Duke M; Tedesco, Rosanna; Ashcraft, Luke W; Yao, Bing; Jiang, Hong; Huang, Jennifer K; Marin, Melchor V; Aroyan, Carrie E; Wang, Jianchao; Ahmed, Seyed; Burgess, Joelle L; Chaudhari, Amita M; Donatelli, Carla A; Darcy, Michael G; Ridgers, Lance H; Newlander, Ken A; Schmidt, Stanley J; Chai, Deping; Colón, Mariela; Zimmerman, Michael N; Lad, Latesh; Sakowicz, Roman; Schauer, Stephen; Belmont, Lisa; Baliga, Ramesh; Pierce, Daniel W; Finer, Jeffrey T; Wang, Zhengping; Morgan, Bradley P; Morgans, David J; Auger, Kurt R; Sung, Chiu-Mei; Carson, Jeff D; Luo, Lusong; Hugger, Erin D; Copeland, Robert A; Sutton, David; Elliott, John D; Jackson, Jeffrey R; Wood, Kenneth W; Dhanak, Dashyant; Bergnes, Gustave; Knight, Steven D.
Affiliation
  • Qian X; Cytokinetics, Inc., 280 E Grand Avenue, South San Francisco, California 94080.
  • McDonald A; Cytokinetics, Inc., 280 E Grand Avenue, South San Francisco, California 94080.
  • Zhou HJ; Cytokinetics, Inc., 280 E Grand Avenue, South San Francisco, California 94080.
  • Adams ND; Oncology R&D, GlaxoSmithKline, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426.
  • Parrish CA; Oncology R&D, GlaxoSmithKline, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426.
  • Duffy KJ; Oncology R&D, GlaxoSmithKline, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426.
  • Fitch DM; Oncology R&D, GlaxoSmithKline, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426.
  • Tedesco R; Oncology R&D, GlaxoSmithKline, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426.
  • Ashcraft LW; Cytokinetics, Inc., 280 E Grand Avenue, South San Francisco, California 94080.
  • Yao B; Cytokinetics, Inc., 280 E Grand Avenue, South San Francisco, California 94080.
  • Jiang H; Cytokinetics, Inc., 280 E Grand Avenue, South San Francisco, California 94080.
  • Huang JK; Cytokinetics, Inc., 280 E Grand Avenue, South San Francisco, California 94080.
  • Marin MV; Cytokinetics, Inc., 280 E Grand Avenue, South San Francisco, California 94080.
  • Aroyan CE; Cytokinetics, Inc., 280 E Grand Avenue, South San Francisco, California 94080.
  • Wang J; Cytokinetics, Inc., 280 E Grand Avenue, South San Francisco, California 94080.
  • Ahmed S; Cytokinetics, Inc., 280 E Grand Avenue, South San Francisco, California 94080.
  • Burgess JL; Oncology R&D, GlaxoSmithKline, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426.
  • Chaudhari AM; Oncology R&D, GlaxoSmithKline, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426.
  • Donatelli CA; Oncology R&D, GlaxoSmithKline, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426.
  • Darcy MG; Oncology R&D, GlaxoSmithKline, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426.
  • Ridgers LH; Oncology R&D, GlaxoSmithKline, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426.
  • Newlander KA; Oncology R&D, GlaxoSmithKline, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426.
  • Schmidt SJ; Oncology R&D, GlaxoSmithKline, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426.
  • Chai D; Oncology R&D, GlaxoSmithKline, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426.
  • Colón M; Oncology R&D, GlaxoSmithKline, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426.
  • Zimmerman MN; Oncology R&D, GlaxoSmithKline, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426.
  • Lad L; Cytokinetics, Inc., 280 E Grand Avenue, South San Francisco, California 94080.
  • Sakowicz R; Cytokinetics, Inc., 280 E Grand Avenue, South San Francisco, California 94080.
  • Schauer S; Cytokinetics, Inc., 280 E Grand Avenue, South San Francisco, California 94080.
  • Belmont L; Cytokinetics, Inc., 280 E Grand Avenue, South San Francisco, California 94080.
  • Baliga R; Cytokinetics, Inc., 280 E Grand Avenue, South San Francisco, California 94080.
  • Pierce DW; Cytokinetics, Inc., 280 E Grand Avenue, South San Francisco, California 94080.
  • Finer JT; Cytokinetics, Inc., 280 E Grand Avenue, South San Francisco, California 94080.
  • Wang Z; Cytokinetics, Inc., 280 E Grand Avenue, South San Francisco, California 94080.
  • Morgan BP; Cytokinetics, Inc., 280 E Grand Avenue, South San Francisco, California 94080.
  • Morgans DJ; Cytokinetics, Inc., 280 E Grand Avenue, South San Francisco, California 94080.
  • Auger KR; Oncology R&D, GlaxoSmithKline, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426.
  • Sung CM; Oncology R&D, GlaxoSmithKline, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426.
  • Carson JD; Oncology R&D, GlaxoSmithKline, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426.
  • Luo L; Oncology R&D, GlaxoSmithKline, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426.
  • Hugger ED; Oncology R&D, GlaxoSmithKline, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426.
  • Copeland RA; Oncology R&D, GlaxoSmithKline, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426.
  • Sutton D; Oncology R&D, GlaxoSmithKline, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426.
  • Elliott JD; Oncology R&D, GlaxoSmithKline, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426.
  • Jackson JR; Oncology R&D, GlaxoSmithKline, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426.
  • Wood KW; Cytokinetics, Inc., 280 E Grand Avenue, South San Francisco, California 94080.
  • Dhanak D; Oncology R&D, GlaxoSmithKline, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426.
  • Bergnes G; Cytokinetics, Inc., 280 E Grand Avenue, South San Francisco, California 94080.
  • Knight SD; Oncology R&D, GlaxoSmithKline, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426.
ACS Med Chem Lett ; 1(1): 30-4, 2010 Apr 08.
Article in En | MEDLINE | ID: mdl-24900171

Full text: 1 Collection: 01-internacional Database: MEDLINE Type of study: Risk_factors_studies Language: En Journal: ACS Med Chem Lett Year: 2010 Document type: Article Country of publication:

Full text: 1 Collection: 01-internacional Database: MEDLINE Type of study: Risk_factors_studies Language: En Journal: ACS Med Chem Lett Year: 2010 Document type: Article Country of publication: