Identification of ligand efficient, fragment-like hits from an HTS library: structure-based virtual screening and docking investigations of 2H- and 3H-pyrazolo tautomers for Aurora kinase A selectivity.
J Comput Aided Mol Des
; 29(1): 89-100, 2015 Jan.
Article
in En
| MEDLINE
| ID: mdl-25344840
Full text:
1
Collection:
01-internacional
Database:
MEDLINE
Main subject:
Structure-Activity Relationship
/
Protein Kinase Inhibitors
/
Drug Evaluation, Preclinical
/
High-Throughput Screening Assays
/
Aurora Kinase A
Type of study:
Diagnostic_studies
/
Prognostic_studies
/
Screening_studies
Limits:
Humans
Language:
En
Journal:
J Comput Aided Mol Des
Journal subject:
BIOLOGIA MOLECULAR
/
ENGENHARIA BIOMEDICA
Year:
2015
Document type:
Article
Affiliation country:
Country of publication: