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Stimulation of cortical bone formation with thienopyrimidine based inhibitors of Notum Pectinacetylesterase.
Tarver, James E; Pabba, Praveen K; Barbosa, Joseph; Han, Qiang; Gardyan, Michael W; Brommage, Robert; Thompson, Andrea Y; Schmidt, James M; Wilson, Alan G E; He, Wei; Lombardo, Victoria K; Carson, Kenneth G.
Affiliation
  • Tarver JE; Lexicon Pharmaceuticals, 350 Carter Road, Princeton, NJ 08540, United States. Electronic address: james.tarver2@gmail.com.
  • Pabba PK; Lexicon Pharmaceuticals, 350 Carter Road, Princeton, NJ 08540, United States.
  • Barbosa J; Lexicon Pharmaceuticals, 350 Carter Road, Princeton, NJ 08540, United States.
  • Han Q; Lexicon Pharmaceuticals, 350 Carter Road, Princeton, NJ 08540, United States.
  • Gardyan MW; Lexicon Pharmaceuticals, 350 Carter Road, Princeton, NJ 08540, United States.
  • Brommage R; Lexicon Pharmaceuticals, 8800 Technology Forest Place, The Woodlands, TX 77381, United States.
  • Thompson AY; Lexicon Pharmaceuticals, 8800 Technology Forest Place, The Woodlands, TX 77381, United States.
  • Schmidt JM; Lexicon Pharmaceuticals, 8800 Technology Forest Place, The Woodlands, TX 77381, United States.
  • Wilson AGE; Lexicon Pharmaceuticals, 8800 Technology Forest Place, The Woodlands, TX 77381, United States.
  • He W; Lexicon Pharmaceuticals, 350 Carter Road, Princeton, NJ 08540, United States.
  • Lombardo VK; Lexicon Pharmaceuticals, 350 Carter Road, Princeton, NJ 08540, United States.
  • Carson KG; Lexicon Pharmaceuticals, 350 Carter Road, Princeton, NJ 08540, United States.
Bioorg Med Chem Lett ; 26(6): 1525-1528, 2016 Mar 15.
Article in En | MEDLINE | ID: mdl-26897593

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Osteogenesis / Pyrimidines / Enzyme Inhibitors / Esterases / Femur Limits: Animals / Humans Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2016 Document type: Article Country of publication:

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Osteogenesis / Pyrimidines / Enzyme Inhibitors / Esterases / Femur Limits: Animals / Humans Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2016 Document type: Article Country of publication: