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Structural Basis for the Selective Binding of Inhibitors to 6-Hydroxymethyl-7,8-dihydropterin Pyrophosphokinase from Staphylococcus aureus and Escherichia coli.
Dennis, Matthew L; Pitcher, Noel P; Lee, Michael D; DeBono, Aaron J; Wang, Zhong-Chang; Harjani, Jitendra R; Rahmani, Raphaël; Cleary, Ben; Peat, Thomas S; Baell, Jonathan B; Swarbrick, James D.
Affiliation
  • Dennis ML; Monash Institute of Pharmaceutical Sciences, Monash University , Parkville, Victoria 3052, Australia.
  • Pitcher NP; CSIRO Biosciences Program , Parkville, Victoria 3052, Australia.
  • Lee MD; Monash Institute of Pharmaceutical Sciences, Monash University , Parkville, Victoria 3052, Australia.
  • DeBono AJ; Monash Institute of Pharmaceutical Sciences, Monash University , Parkville, Victoria 3052, Australia.
  • Wang ZC; Monash Institute of Pharmaceutical Sciences, Monash University , Parkville, Victoria 3052, Australia.
  • Harjani JR; Monash Institute of Pharmaceutical Sciences, Monash University , Parkville, Victoria 3052, Australia.
  • Rahmani R; State Key Laboratory of Pharmaceutical Biotechnology, Nanjing University , Nanjing 210093, People's Republic of China.
  • Cleary B; Monash Institute of Pharmaceutical Sciences, Monash University , Parkville, Victoria 3052, Australia.
  • Peat TS; Monash Institute of Pharmaceutical Sciences, Monash University , Parkville, Victoria 3052, Australia.
  • Baell JB; Monash Institute of Pharmaceutical Sciences, Monash University , Parkville, Victoria 3052, Australia.
  • Swarbrick JD; CSIRO Biosciences Program , Parkville, Victoria 3052, Australia.
J Med Chem ; 59(11): 5248-63, 2016 06 09.
Article in En | MEDLINE | ID: mdl-27094768

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Staphylococcus aureus / Diphosphotransferases / Enzyme Inhibitors / Escherichia coli Language: En Journal: J Med Chem Journal subject: QUIMICA Year: 2016 Document type: Article Affiliation country: Country of publication:

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Staphylococcus aureus / Diphosphotransferases / Enzyme Inhibitors / Escherichia coli Language: En Journal: J Med Chem Journal subject: QUIMICA Year: 2016 Document type: Article Affiliation country: Country of publication: