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1,4-Substituted Triazoles as Nonsteroidal Anti-Androgens for Prostate Cancer Treatment.
Ferroni, Claudia; Pepe, Antonella; Kim, Yeong Sang; Lee, Sunmin; Guerrini, Andrea; Parenti, Marco Daniele; Tesei, Anna; Zamagni, Alice; Cortesi, Michela; Zaffaroni, Nadia; De Cesare, Michelandrea; Beretta, Giovanni Luca; Trepel, Jane B; Malhotra, Sanjay V; Varchi, Greta.
Affiliation
  • Ferroni C; Institute for the Organic Synthesis and Photoreactivity, Italian National Research Council , Via Gobetti 101, 40129 Bologna, Italy.
  • Pepe A; Purdue Center for Cancer Research , 720 Clinic Drive, West Lafayette, Indiana 47907, United States.
  • Kim YS; Center for Cancer Research, National Cancer Institute, National Institutes of Health , Building 10, Magnuson CC, Bethesda, Maryland 20892, United States.
  • Lee S; Center for Cancer Research, National Cancer Institute, National Institutes of Health , Building 10, Magnuson CC, Bethesda, Maryland 20892, United States.
  • Guerrini A; Institute for the Organic Synthesis and Photoreactivity, Italian National Research Council , Via Gobetti 101, 40129 Bologna, Italy.
  • Parenti MD; Institute for the Organic Synthesis and Photoreactivity, Italian National Research Council , Via Gobetti 101, 40129 Bologna, Italy.
  • Tesei A; Biosciences Laboratory, Istituto Scientifico Romagnolo per lo Studio e la Cura dei Tumori (IRST), IRCCS , Via P. Maroncelli, 40, 47014 Meldola, Forlì Italy.
  • Zamagni A; Biosciences Laboratory, Istituto Scientifico Romagnolo per lo Studio e la Cura dei Tumori (IRST), IRCCS , Via P. Maroncelli, 40, 47014 Meldola, Forlì Italy.
  • Cortesi M; Biosciences Laboratory, Istituto Scientifico Romagnolo per lo Studio e la Cura dei Tumori (IRST), IRCCS , Via P. Maroncelli, 40, 47014 Meldola, Forlì Italy.
  • Zaffaroni N; Fondazione IRCCS Istituto Tumori Milano , Via Amadeo, 42, 20133 Milano, Italy.
  • De Cesare M; Fondazione IRCCS Istituto Tumori Milano , Via Amadeo, 42, 20133 Milano, Italy.
  • Beretta GL; Fondazione IRCCS Istituto Tumori Milano , Via Amadeo, 42, 20133 Milano, Italy.
  • Trepel JB; Center for Cancer Research, National Cancer Institute, National Institutes of Health , Building 10, Magnuson CC, Bethesda, Maryland 20892, United States.
  • Malhotra SV; Department of Radiation Oncology, Division of Radiation and Cancer Biology, Stanford University School of Medicine , Stanford, California 94304, United States.
  • Varchi G; Institute for the Organic Synthesis and Photoreactivity, Italian National Research Council , Via Gobetti 101, 40129 Bologna, Italy.
J Med Chem ; 60(7): 3082-3093, 2017 04 13.
Article in En | MEDLINE | ID: mdl-28272894

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Prostate / Prostatic Neoplasms / Triazoles / Nonsteroidal Anti-Androgens Limits: Animals / Humans / Male Language: En Journal: J Med Chem Journal subject: QUIMICA Year: 2017 Document type: Article Affiliation country: Country of publication:

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Prostate / Prostatic Neoplasms / Triazoles / Nonsteroidal Anti-Androgens Limits: Animals / Humans / Male Language: En Journal: J Med Chem Journal subject: QUIMICA Year: 2017 Document type: Article Affiliation country: Country of publication: