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ERE-dependent transcription and cell proliferation: Independency of these two processes mediated by the introduction of a sulfone function into the weak estrogen estrothiazine.
Jacquot, Yves; Spaggiari, Dany; Schappler, Julie; Lesniewska, Eric; Rudaz, Serge; Leclercq, Guy.
Affiliation
  • Jacquot Y; Sorbonne University - UPMC Univ Paris 06, Ecole Normale Supérieure, PSL Research University, Département de Chimie, CNRS UMR 7203 LBM, 4 Place Jussieu, 75005 Paris, France. Electronic address: yves.jacquot@upmc.fr.
  • Spaggiari D; Section des Sciences Pharmaceutiques (EPGL), University of Geneva, University of Lausanne, rue Michel Servet 1, 1211 Geneva 4, Switzerland.
  • Schappler J; Section des Sciences Pharmaceutiques (EPGL), University of Geneva, University of Lausanne, rue Michel Servet 1, 1211 Geneva 4, Switzerland.
  • Lesniewska E; ICB, CNRS UMR 6303, University de Bourgogne Franche-Comté, 9, avenue Savary, 21078 Dijon, France.
  • Rudaz S; Section des Sciences Pharmaceutiques (EPGL), University of Geneva, University of Lausanne, rue Michel Servet 1, 1211 Geneva 4, Switzerland.
  • Leclercq G; Laboratory J.C. Heuson de Cancérologie Mammaire, Institut Jules Bordet, 1, rue Héger Bordet, Brussels 1000, Belgium. Electronic address: guy.leclercq@ulb.ac.be.
Eur J Pharm Sci ; 109: 169-181, 2017 Nov 15.
Article in En | MEDLINE | ID: mdl-28754571

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Sulfones / Coumarins / Estrogen Receptor alpha / Estrogens Type of study: Prognostic_studies Limits: Humans Language: En Journal: Eur J Pharm Sci Journal subject: FARMACIA / FARMACOLOGIA / QUIMICA Year: 2017 Document type: Article Country of publication:

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Sulfones / Coumarins / Estrogen Receptor alpha / Estrogens Type of study: Prognostic_studies Limits: Humans Language: En Journal: Eur J Pharm Sci Journal subject: FARMACIA / FARMACOLOGIA / QUIMICA Year: 2017 Document type: Article Country of publication: