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Molecular modeling and biological studies show that some µ-opioid receptor agonists might elicit analgesia acting as MMP-9 inhibitors.
Ronsisvalle, Simone; Spadaro, Angelo; Tomasello, Barbara; Basile, Livia; Panarello, Federica; Franchini, Silvia; Renis, Marcella; Guccione, Salvatore; Crascì, Lucia; Panico, Anna Maria.
Affiliation
  • Ronsisvalle S; Department of Drug Sciences, Medicinal Chemistry Section, University of Catania, Viale A Doria 6, I-95125 Catania, Italy.
  • Spadaro A; Department of Drug Sciences, Medicinal Chemistry Section, University of Catania, Viale A Doria 6, I-95125 Catania, Italy.
  • Tomasello B; Department of Drug Sciences, Biochemistry Section, University of Catania, Viale A Doria 6, I-95125 Catania, Italy.
  • Basile L; Department of Drug Sciences, Medicinal Chemistry Section, University of Catania, Viale A Doria 6, I-95125 Catania, Italy.
  • Panarello F; Department of Drug Sciences, Medicinal Chemistry Section, University of Catania, Viale A Doria 6, I-95125 Catania, Italy.
  • Franchini S; Dipartimento di Scienze della Vita, Universita' di Modena e Reggio Emilia, Via Campi 103, I-41125 Modena, Italy.
  • Renis M; Department of Drug Sciences, Biochemistry Section, University of Catania, Viale A Doria 6, I-95125 Catania, Italy.
  • Guccione S; Department of Drug Sciences, Medicinal Chemistry Section, University of Catania, Viale A Doria 6, I-95125 Catania, Italy.
  • Crascì L; Department of Drug Sciences, Medicinal Chemistry Section, University of Catania, Viale A Doria 6, I-95125 Catania, Italy.
  • Panico AM; Department of Drug Sciences, Medicinal Chemistry Section, University of Catania, Viale A Doria 6, I-95125 Catania, Italy.
Future Med Chem ; 11(11): 1245-1258, 2019 06.
Article in En | MEDLINE | ID: mdl-30974972

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Benzomorphans / Receptors, Opioid, mu / Matrix Metalloproteinase 9 / Matrix Metalloproteinase Inhibitors / Analgesics Limits: Humans Language: En Journal: Future Med Chem Year: 2019 Document type: Article Affiliation country: Country of publication:

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Benzomorphans / Receptors, Opioid, mu / Matrix Metalloproteinase 9 / Matrix Metalloproteinase Inhibitors / Analgesics Limits: Humans Language: En Journal: Future Med Chem Year: 2019 Document type: Article Affiliation country: Country of publication: