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Structural Basis and Kinetic Pathway of RBM39 Recruitment to DCAF15 by a Sulfonamide Molecular Glue E7820.
Du, Xinlin; Volkov, Oleg A; Czerwinski, Robert M; Tan, HuiLing; Huerta, Carlos; Morton, Emily R; Rizzi, Jim P; Wehn, Paul M; Xu, Rui; Nijhawan, Deepak; Wallace, Eli M.
Affiliation
  • Du X; Peloton Therapeutics, Dallas, Texas, a Subsidiary of Merck & Co., Inc., Kenilworth, NJ 07033, USA. Electronic address: xinlin.du@merck.com.
  • Volkov OA; Peloton Therapeutics, Dallas, Texas, a Subsidiary of Merck & Co., Inc., Kenilworth, NJ 07033, USA.
  • Czerwinski RM; Peloton Therapeutics, Dallas, Texas, a Subsidiary of Merck & Co., Inc., Kenilworth, NJ 07033, USA.
  • Tan H; Peloton Therapeutics, Dallas, Texas, a Subsidiary of Merck & Co., Inc., Kenilworth, NJ 07033, USA.
  • Huerta C; Peloton Therapeutics, Dallas, Texas, a Subsidiary of Merck & Co., Inc., Kenilworth, NJ 07033, USA.
  • Morton ER; Peloton Therapeutics, Dallas, Texas, a Subsidiary of Merck & Co., Inc., Kenilworth, NJ 07033, USA.
  • Rizzi JP; Peloton Therapeutics, Dallas, Texas, a Subsidiary of Merck & Co., Inc., Kenilworth, NJ 07033, USA.
  • Wehn PM; Peloton Therapeutics, Dallas, Texas, a Subsidiary of Merck & Co., Inc., Kenilworth, NJ 07033, USA.
  • Xu R; Peloton Therapeutics, Dallas, Texas, a Subsidiary of Merck & Co., Inc., Kenilworth, NJ 07033, USA.
  • Nijhawan D; Departments of Biochemistry and Internal Medicine, University of Texas, Southwestern Medical Center, Dallas, TX 75390, USA.
  • Wallace EM; Peloton Therapeutics, Dallas, Texas, a Subsidiary of Merck & Co., Inc., Kenilworth, NJ 07033, USA.
Structure ; 27(11): 1625-1633.e3, 2019 11 05.
Article in En | MEDLINE | ID: mdl-31693911

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Sulfonamides / RNA-Binding Proteins / Intracellular Signaling Peptides and Proteins / Indoles Limits: Humans Language: En Journal: Structure Journal subject: BIOLOGIA MOLECULAR / BIOQUIMICA / BIOTECNOLOGIA Year: 2019 Document type: Article Country of publication:

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Sulfonamides / RNA-Binding Proteins / Intracellular Signaling Peptides and Proteins / Indoles Limits: Humans Language: En Journal: Structure Journal subject: BIOLOGIA MOLECULAR / BIOQUIMICA / BIOTECNOLOGIA Year: 2019 Document type: Article Country of publication: