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3-Bromopyruvate as a potent covalently reversible inhibitor of New Delhi metallo-ß-lactamase-1 (NDM-1).
Kang, Peng-Wei; Su, Jian-Peng; Sun, Le-Yun; Gao, Han; Yang, Ke-Wu.
Affiliation
  • Kang PW; Key Laboratory of Synthetic and Natural Functional Molecule Chemistry of Ministry of Education, College of Chemistry and Materials Science, Northwest University, 1 Xuefu Avenue, Xi'an 710127, PR China.
  • Su JP; Key Laboratory of Synthetic and Natural Functional Molecule Chemistry of Ministry of Education, College of Chemistry and Materials Science, Northwest University, 1 Xuefu Avenue, Xi'an 710127, PR China.
  • Sun LY; Key Laboratory of Synthetic and Natural Functional Molecule Chemistry of Ministry of Education, College of Chemistry and Materials Science, Northwest University, 1 Xuefu Avenue, Xi'an 710127, PR China.
  • Gao H; Key Laboratory of Synthetic and Natural Functional Molecule Chemistry of Ministry of Education, College of Chemistry and Materials Science, Northwest University, 1 Xuefu Avenue, Xi'an 710127, PR China.
  • Yang KW; Key Laboratory of Synthetic and Natural Functional Molecule Chemistry of Ministry of Education, College of Chemistry and Materials Science, Northwest University, 1 Xuefu Avenue, Xi'an 710127, PR China. Electronic address: kwyang@nwu.edu.cn.
Eur J Pharm Sci ; 142: 105161, 2020 Jan 15.
Article in En | MEDLINE | ID: mdl-31751778

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Pyruvates / Beta-Lactamases / Anti-Bacterial Agents Limits: Animals Language: En Journal: Eur J Pharm Sci Journal subject: FARMACIA / FARMACOLOGIA / QUIMICA Year: 2020 Document type: Article

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Pyruvates / Beta-Lactamases / Anti-Bacterial Agents Limits: Animals Language: En Journal: Eur J Pharm Sci Journal subject: FARMACIA / FARMACOLOGIA / QUIMICA Year: 2020 Document type: Article