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Thienopyrimidine Derivatives as GPR55 Receptor Antagonists: Insight into Structure-Activity Relationship.
Figuerola-Asencio, Laura; Morales, Paula; Zhao, Pingwei; Hurst, Dow P; Sayed, Sommayah S; Colón, Katsuya L; Gómez-Cañas, María; Fernández-Ruiz, Javier; Croatt, Mitchell P; Reggio, Patricia H; Abood, Mary E; Jagerovic, Nadine.
Affiliation
  • Figuerola-Asencio L; Instituto de Química Médica, Consejo Superior de Investigaciones Científicas, 28006Madrid, Spain.
  • Morales P; Instituto de Química Médica, Consejo Superior de Investigaciones Científicas, 28006Madrid, Spain.
  • Zhao P; Center for Substance Abuse Research, Temple University, Philadelphia, Pennsylvania19122, United States.
  • Hurst DP; Center for Drug Discovery, Department of Chemistry and Biochemistry, University North Carolina, Greensboro, North Carolina27599, United States.
  • Sayed SS; Center for Drug Discovery, Department of Chemistry and Biochemistry, University North Carolina, Greensboro, North Carolina27599, United States.
  • Colón KL; Center for Drug Discovery, Department of Chemistry and Biochemistry, University North Carolina, Greensboro, North Carolina27599, United States.
  • Gómez-Cañas M; Department of Biochemistry and Molecular Biology, Faculty of Medicine, Complutense University, CIBERNED and IRYCIS, 28040Madrid, Spain.
  • Fernández-Ruiz J; Department of Biochemistry and Molecular Biology, Faculty of Medicine, Complutense University, CIBERNED and IRYCIS, 28040Madrid, Spain.
  • Croatt MP; Center for Drug Discovery, Department of Chemistry and Biochemistry, University North Carolina, Greensboro, North Carolina27599, United States.
  • Reggio PH; Center for Drug Discovery, Department of Chemistry and Biochemistry, University North Carolina, Greensboro, North Carolina27599, United States.
  • Abood ME; Center for Substance Abuse Research, Temple University, Philadelphia, Pennsylvania19122, United States.
  • Jagerovic N; Instituto de Química Médica, Consejo Superior de Investigaciones Científicas, 28006Madrid, Spain.
ACS Med Chem Lett ; 14(1): 18-25, 2023 Jan 12.
Article in En | MEDLINE | ID: mdl-36655130

Full text: 1 Collection: 01-internacional Database: MEDLINE Language: En Journal: ACS Med Chem Lett Year: 2023 Document type: Article Affiliation country:

Full text: 1 Collection: 01-internacional Database: MEDLINE Language: En Journal: ACS Med Chem Lett Year: 2023 Document type: Article Affiliation country: