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Identification of Novel Compounds Inhibiting the Kinase Activity of the CDK5/p25 Complex via Direct Binding to p25.
Jabeur, Riheb; Corbel, Caroline; Loyer, Pascal; Le Parc, Annabelle; Le Grand, Adélaide; Comte, Arnaud; Bach, Stéphane; André-Leroux, Gwenaëlle; Sire, Olivier; Ben Mansour, Hedi; Le Tilly, Véronique.
Affiliation
  • Jabeur R; IRDL UMR CNRS 6027, Université Bretagne Sud, 56017 Vannes, France.
  • Corbel C; Research Unit of Analysis and Process Applied on the Environment─APAE UR17ES32, Higher Institute of Applied Sciences and Technology, Mahdia, University of Monastir, TN5121 Monastir, Tunisia.
  • Loyer P; IRDL UMR CNRS 6027, Université Bretagne Sud, 56017 Vannes, France.
  • Le Parc A; Univ Rennes, INSERM, INRAE, Institut NuMeCan (Nutrition, Metabolisms and Cancer) UMR-A 1341, UMR-S 1241, F-35000 Rennes, France.
  • Le Grand A; Aspen Pharmacare, 76960 Notre-Dame-de-Bondeville, France.
  • Comte A; IRDL UMR CNRS 6027, Université Bretagne Sud, 56017 Vannes, France.
  • Bach S; Compound Library, ICBMS UMR 5246 CNRS-Université Claude Bernard Lyon 1, Université de Lyon, 69622 Villeurbanne, France.
  • André-Leroux G; Sorbonne Université, CNRS, UMR8227, Integrative Biology of Marine Models Laboratory (LBI2M), Station Biologique de Roscoff, 29680 Roscoff, France.
  • Sire O; Sorbonne Université, CNRS, FR2424, Plateforme de criblage KISSf (Kinase Inhibitor Specialized Screening facility), Station Biologique de Roscoff, 29680 Roscoff, France.
  • Ben Mansour H; Centre of Excellence for Pharmaceutical Sciences, North-West University, Private Bag X6001, 2520 Potchefstroom, South Africa.
  • Le Tilly V; Université Paris-Sac, INRAE, MaIAGElay, 78350 Jouy-en-Josas, France.
Biochemistry ; 62(9): 1452-1463, 2023 05 02.
Article in En | MEDLINE | ID: mdl-37074084

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Breast Neoplasms / Alzheimer Disease Type of study: Diagnostic_studies Limits: Female / Humans Language: En Journal: Biochemistry Year: 2023 Document type: Article Affiliation country:

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Breast Neoplasms / Alzheimer Disease Type of study: Diagnostic_studies Limits: Female / Humans Language: En Journal: Biochemistry Year: 2023 Document type: Article Affiliation country: