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A Systematic Survey of Reversibly Covalent Dipeptidyl Inhibitors of the SARS-CoV-2 Main Protease.
Geng, Zhi Zachary; Atla, Sandeep; Shaabani, Namir; Vulupala, Veerabhadra; Yang, Kai S; Alugubelli, Yugendar R; Khatua, Kaustav; Chen, Peng-Hsun; Xiao, Jing; Blankenship, Lauren R; Ma, Xinyu R; Vatansever, Erol C; Cho, Chia-Chuan D; Ma, Yuying; Allen, Robert; Ji, Henry; Xu, Shiqing; Liu, Wenshe Ray.
Affiliation
  • Geng ZZ; Department of Chemistry, Texas A&M Drug Discovery Laboratory, Texas A&M University, College Station, Texas 77843, United States.
  • Atla S; Department of Chemistry, Texas A&M Drug Discovery Laboratory, Texas A&M University, College Station, Texas 77843, United States.
  • Shaabani N; Sorrento Therapeutics, Inc. San Diego, California 92121, United States.
  • Vulupala V; Department of Chemistry, Texas A&M Drug Discovery Laboratory, Texas A&M University, College Station, Texas 77843, United States.
  • Yang KS; Department of Chemistry, Texas A&M Drug Discovery Laboratory, Texas A&M University, College Station, Texas 77843, United States.
  • Alugubelli YR; Department of Chemistry, Texas A&M Drug Discovery Laboratory, Texas A&M University, College Station, Texas 77843, United States.
  • Khatua K; Department of Chemistry, Texas A&M Drug Discovery Laboratory, Texas A&M University, College Station, Texas 77843, United States.
  • Chen PH; Department of Chemistry, Texas A&M Drug Discovery Laboratory, Texas A&M University, College Station, Texas 77843, United States.
  • Xiao J; Department of Chemistry, Texas A&M Drug Discovery Laboratory, Texas A&M University, College Station, Texas 77843, United States.
  • Blankenship LR; Department of Chemistry, Texas A&M Drug Discovery Laboratory, Texas A&M University, College Station, Texas 77843, United States.
  • Ma XR; Department of Chemistry, Texas A&M Drug Discovery Laboratory, Texas A&M University, College Station, Texas 77843, United States.
  • Vatansever EC; Department of Chemistry, Texas A&M Drug Discovery Laboratory, Texas A&M University, College Station, Texas 77843, United States.
  • Cho CD; Department of Chemistry, Texas A&M Drug Discovery Laboratory, Texas A&M University, College Station, Texas 77843, United States.
  • Ma Y; Department of Chemistry, Texas A&M Drug Discovery Laboratory, Texas A&M University, College Station, Texas 77843, United States.
  • Allen R; Sorrento Therapeutics, Inc. San Diego, California 92121, United States.
  • Ji H; Sorrento Therapeutics, Inc. San Diego, California 92121, United States.
  • Xu S; Department of Chemistry, Texas A&M Drug Discovery Laboratory, Texas A&M University, College Station, Texas 77843, United States.
  • Liu WR; Department of Pharmaceutical Sciences, Irma Lerma Rangel College of Pharmacy, Texas A&M University, College Station, Texas 77843, United States.
J Med Chem ; 66(16): 11040-11055, 2023 08 24.
Article in En | MEDLINE | ID: mdl-37561993

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: COVID-19 Limits: Humans Language: En Journal: J Med Chem Journal subject: QUIMICA Year: 2023 Document type: Article Affiliation country:

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: COVID-19 Limits: Humans Language: En Journal: J Med Chem Journal subject: QUIMICA Year: 2023 Document type: Article Affiliation country: