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Structural Optimization of Decoy Oligonucleotide-Based PROTAC That Degrades the Estrogen Receptor.
Naganuma, Miyako; Ohoka, Nobumichi; Tsuji, Genichiro; Inoue, Takao; Naito, Mikihiko; Demizu, Yosuke.
Affiliation
  • Naganuma M; Division of Organic Chemistry, National Institute of Health Sciences, Kanagawa 210-9501, Japan.
  • Ohoka N; Graduate School of Medical Life Science, Yokohama City University, Kanagawa 236-0027, Japan.
  • Tsuji G; Division of Molecular Target and Gene Therapy Products, National Institute of Health Sciences, Kanagawa 210-9501, Japan.
  • Inoue T; Division of Organic Chemistry, National Institute of Health Sciences, Kanagawa 210-9501, Japan.
  • Naito M; Division of Molecular Target and Gene Therapy Products, National Institute of Health Sciences, Kanagawa 210-9501, Japan.
  • Demizu Y; Laboratory of Targeted Protein Degradation, Graduate School of Pharmaceutical Sciences, The University of Tokyo, Tokyo 110-0033, Japan.
Bioconjug Chem ; 34(10): 1780-1788, 2023 10 18.
Article in En | MEDLINE | ID: mdl-37736001

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Receptors, Estrogen / Estrogen Receptor alpha / Proteolysis Targeting Chimera Type of study: Prognostic_studies Limits: Humans Language: En Journal: Bioconjug Chem Journal subject: BIOQUIMICA Year: 2023 Document type: Article Affiliation country: Country of publication:

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Receptors, Estrogen / Estrogen Receptor alpha / Proteolysis Targeting Chimera Type of study: Prognostic_studies Limits: Humans Language: En Journal: Bioconjug Chem Journal subject: BIOQUIMICA Year: 2023 Document type: Article Affiliation country: Country of publication: