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TMSOTf-Promoted Cyclization of Indole-2-methyl-α-aminoketones: Access to 4-Aryl-Substituted ß-Carbolines.
Yang, Xin-Yu; Yang, Jin-Ming; Wu, Bin.
Affiliation
  • Yang XY; School of Pharmaceutical Sciences, South-Central Minzu University, Wuhan 430074, China.
  • Yang JM; School of Pharmaceutical Sciences, South-Central Minzu University, Wuhan 430074, China.
  • Wu B; School of Pharmaceutical Sciences, South-Central Minzu University, Wuhan 430074, China.
Org Lett ; 26(5): 1105-1109, 2024 Feb 09.
Article in En | MEDLINE | ID: mdl-38289176
ABSTRACT
An efficient method to construct 4-aryl-substituted ß-carbolines from indole-2-methyl-α-aminoketones via a TMSOTf-promoted annulation reaction was reported. High yield along with wide substrate scope and functional group tolerance make this reaction applicable to build various highly potential bioactive ß-carboline derivatives.
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Full text: 1 Collection: 01-internacional Database: MEDLINE Language: En Journal: Org Lett Journal subject: BIOQUIMICA Year: 2024 Document type: Article Affiliation country: Country of publication:
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Full text: 1 Collection: 01-internacional Database: MEDLINE Language: En Journal: Org Lett Journal subject: BIOQUIMICA Year: 2024 Document type: Article Affiliation country: Country of publication: