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Design of hypoxia-targeting protein tyrosine kinase inhibitor using an innovative pharmacophore 2-methylene-4-cyclopentene-1,3-dione.
Hori, Hitoshi; Nagasawa, Hideko; Uto, Yoshihiro; Ohkura, Kazuto; Kirk, Kenneth L; Uehara, Yoshimasa; Shimamura, Mariko.
Affiliation
  • Hori H; Department of Biological Science and Technology, Faculty of Engineering, The University of Tokushima, Minamijosanjimacho-2, Tokushima 770-8506, Japan. hori@bio.tokushima-u.ac.jp
Biochim Biophys Acta ; 1697(1-2): 29-38, 2004 Mar 11.
Article in En | MEDLINE | ID: mdl-15023348
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Collection: 01-internacional Database: MEDLINE Main subject: Protein-Tyrosine Kinases / Cell Hypoxia / Cyclopentanes / Enzyme Inhibitors Limits: Animals / Humans Language: En Journal: Biochim Biophys Acta Year: 2004 Document type: Article Affiliation country: Japón Country of publication: Países Bajos
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Collection: 01-internacional Database: MEDLINE Main subject: Protein-Tyrosine Kinases / Cell Hypoxia / Cyclopentanes / Enzyme Inhibitors Limits: Animals / Humans Language: En Journal: Biochim Biophys Acta Year: 2004 Document type: Article Affiliation country: Japón Country of publication: Países Bajos