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Synthesis and structure-activity relationships of novel IKK-beta inhibitors. Part 3: Orally active anti-inflammatory agents.
Murata, Toshiki; Shimada, Mitsuyuki; Sakakibara, Sachiko; Yoshino, Takashi; Masuda, Tsutomu; Shintani, Takuya; Sato, Hiroki; Koriyama, Yuji; Fukushima, Keiko; Nunami, Noriko; Yamauchi, Megumi; Fuchikami, Kinji; Komura, Hiroshi; Watanabe, Akihiko; Ziegelbauer, Karl B; Bacon, Kevin B; Lowinger, Timothy B.
Affiliation
  • Murata T; Department of Chemistry, Research Center Kyoto, Bayer Yakuhin Ltd., Kizu, Soraku, Kyoto 619-0216, Japan. muratato@kcn.ne.jp
Bioorg Med Chem Lett ; 14(15): 4019-22, 2004 Aug 02.
Article in En | MEDLINE | ID: mdl-15225718
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Collection: 01-internacional Database: MEDLINE Main subject: Pyridines / Protein Serine-Threonine Kinases / Anti-Inflammatory Agents Limits: Animals / Humans Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2004 Document type: Article Affiliation country: Japón Country of publication: Reino Unido
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Collection: 01-internacional Database: MEDLINE Main subject: Pyridines / Protein Serine-Threonine Kinases / Anti-Inflammatory Agents Limits: Animals / Humans Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2004 Document type: Article Affiliation country: Japón Country of publication: Reino Unido