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Synthetic muO-conotoxin MrVIB blocks TTX-resistant sodium channel NaV1.8 and has a long-lasting analgesic activity.
Bulaj, Grzegorz; Zhang, Min-Min; Green, Brad R; Fiedler, Brian; Layer, Richard T; Wei, Sue; Nielsen, Jacob S; Low, Scott J; Klein, Brian D; Wagstaff, John D; Chicoine, Linda; Harty, T Patrick; Terlau, Heinrich; Yoshikami, Doju; Olivera, Baldomero M.
Affiliation
  • Bulaj G; Department of Biology, The University of Utah, Salt Lake City, Utah 84112, USA. bulaj@biology.utah.edu
Biochemistry ; 45(23): 7404-14, 2006 Jun 13.
Article in En | MEDLINE | ID: mdl-16752929
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Collection: 01-internacional Database: MEDLINE Main subject: Tetrodotoxin / Conotoxins / Analgesics / Nerve Tissue Proteins Limits: Animals Language: En Journal: Biochemistry Year: 2006 Document type: Article Affiliation country: Estados Unidos Country of publication: Estados Unidos
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Collection: 01-internacional Database: MEDLINE Main subject: Tetrodotoxin / Conotoxins / Analgesics / Nerve Tissue Proteins Limits: Animals Language: En Journal: Biochemistry Year: 2006 Document type: Article Affiliation country: Estados Unidos Country of publication: Estados Unidos