Potent nonpeptide antagonists of the bradykinin B1 receptor: structure-activity relationship studies with novel diaminochroman carboxamides.

Biswas, Kaustav; Li, Aiwen; Chen, Jian Jeffrey; D'Amico, Derin C; Fotsch, Christopher; Han, Nianhe; Human, Jason; Liu, Qingyian; Norman, Mark H; Riahi, Bobby; Yuan, Chester; Suzuki, Hideo; Mareska, David A; Zhan, James; Clarke, David E; Toro, Andras; Groneberg, Robert D; Burgess, Laurence E; Lester-Zeiner, Dianna; Biddlecome, Gloria; Manning, Barton H; Arik, Leyla; Dong, Hong; Huang, Ming; Kamassah, Augustus; Loeloff, Richard; Sun, Hong; Hsieh, Feng-Yin; Kumar, Gondi; Ng, Gordon Y; Hungate, Randall W; Askew, Benny C; Johnson, Eileen

Biswas, Kaustav; Li, Aiwen; Chen, Jian Jeffrey; D'Amico, Derin C; Fotsch, Christopher; Han, Nianhe; Human, Jason; Liu, Qingyian; Norman, Mark H; Riahi, Bobby; Yuan, Chester; Suzuki, Hideo; Mareska, David A; Zhan, James; Clarke, David E; Toro, Andras; Groneberg, Robert D; Burgess, Laurence E; Lester-Zeiner, Dianna; Biddlecome, Gloria; Manning, Barton H; Arik, Leyla; Dong, Hong; Huang, Ming; Kamassah, Augustus; Loeloff, Richard; Sun, Hong; Hsieh, Feng-Yin; Kumar, Gondi; Ng, Gordon Y; Hungate, Randall W; Askew, Benny C; Johnson, Eileen.

Affiliation

Biswas K; Department of Chemistry Research and Discovery, Amgen Inc., One Amgen Center Drive, Thousand Oaks, California 91320, USA. kbiswas@amgen.com

J Med Chem ; 50(9): 2200-12, 2007 May 03.

Article in En | MEDLINE | ID: mdl-17408249

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Collection: 01-internacional Database: MEDLINE Main subject: Sulfonamides / Benzopyrans / Chromans / Bradykinin B1 Receptor Antagonists / Amides / Analgesics Type of study: Guideline / Prognostic_studies Limits: Animals / Humans / Male Language: En Journal: J Med Chem Journal subject: QUIMICA Year: 2007 Document type: Article Affiliation country: Estados Unidos Country of publication: Estados Unidos

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