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Atropisomeric 8-arylchromen-4-ones exhibit enantioselective inhibition of the DNA-dependent protein kinase (DNA-PK).
Cano, Céline; Golding, Bernard T; Haggerty, Karen; Hardcastle, Ian R; Peacock, Marcus; Griffin, Roger J.
Affiliation
  • Cano C; Northern Institute for Cancer Research, School of Chemistry, Bedson Building, Newcastle University, Newcastle upon Tyne, United KingdomNE1 7RU. celine.cano@ncl.ac.uk
Org Biomol Chem ; 8(8): 1922-8, 2010 Apr 21.
Article in En | MEDLINE | ID: mdl-20449499

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Thiophenes / Protein Kinase Inhibitors / DNA-Activated Protein Kinase Language: En Journal: Org Biomol Chem Journal subject: BIOQUIMICA / QUIMICA Year: 2010 Document type: Article Country of publication: Reino Unido

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Thiophenes / Protein Kinase Inhibitors / DNA-Activated Protein Kinase Language: En Journal: Org Biomol Chem Journal subject: BIOQUIMICA / QUIMICA Year: 2010 Document type: Article Country of publication: Reino Unido