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Synthesis and evaluation of 2-phenyl-1,4-butanediamine-based CCR5 antagonists for the treatment of HIV-1.
Tallant, Matthew D; Duan, Maosheng; Freeman, George A; Ferris, Robert G; Edelstein, Mark P; Kazmierski, Wieslaw M; Wheelan, Pat J.
Affiliation
  • Tallant MD; Department of Chemistry, GlaxoSmithKline, Research Triangle Park, NC 27709, USA. matthew.d.tallant@gsk.com
Bioorg Med Chem Lett ; 21(5): 1394-8, 2011 Mar 01.
Article in En | MEDLINE | ID: mdl-21292480

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Putrescine / Anti-HIV Agents / CCR5 Receptor Antagonists Limits: Animals Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2011 Document type: Article Affiliation country: Estados Unidos

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Putrescine / Anti-HIV Agents / CCR5 Receptor Antagonists Limits: Animals Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2011 Document type: Article Affiliation country: Estados Unidos