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Discovery of a Potent, Injectable Inhibitor of Aurora Kinases Based on the Imidazo-[1,2-a]-Pyrazine Core.
Yu, Tao; Tagat, Jayaram R; Kerekes, Angela D; Doll, Ronald J; Zhang, Yonglian; Xiao, Yushi; Esposite, Sara; Belanger, David B; Curran, Patrick J; Mandal, Amit K; Siddiqui, M Arshad; Shih, Neng-Yang; Basso, Andrea D; Liu, Ming; Gray, Kimberly; Tevar, Seema; Jones, Jennifer; Lee, Suining; Liang, Lianzhu; Ponery, Samad; Smith, Elizabeth B; Hruza, Alan; Voigt, Johannes; Ramanathan, Lata; Prosise, Winifred; Hu, Mengwei.
Affiliation
  • Yu T; Departments of Chemical Research.
  • Tagat JR; Departments of Chemical Research.
  • Kerekes AD; Departments of Chemical Research.
  • Doll RJ; Departments of Chemical Research.
  • Zhang Y; Departments of Chemical Research.
  • Xiao Y; Departments of Chemical Research.
  • Esposite S; Departments of Chemical Research.
  • Belanger DB; Department of Chemical Research.
  • Curran PJ; Department of Chemical Research.
  • Mandal AK; Department of Chemical Research.
  • Siddiqui MA; Department of Chemical Research.
  • Shih NY; Department of Chemical Research.
  • Basso AD; Oncology.
  • Liu M; Oncology.
  • Gray K; Oncology.
  • Tevar S; Oncology.
  • Jones J; Oncology.
  • Lee S; Oncology.
  • Liang L; Oncology.
  • Ponery S; Oncology.
  • Smith EB; Oncology.
  • Hruza A; Structural Chemistry.
  • Voigt J; Structural Chemistry.
  • Ramanathan L; Structural Chemistry.
  • Prosise W; Structural Chemistry.
  • Hu M; Pharmaceutical Sciences.
ACS Med Chem Lett ; 1(5): 214-8, 2010 Aug 12.
Article in En | MEDLINE | ID: mdl-24900197

Full text: 1 Collection: 01-internacional Database: MEDLINE Language: En Journal: ACS Med Chem Lett Year: 2010 Document type: Article Country of publication: Estados Unidos

Full text: 1 Collection: 01-internacional Database: MEDLINE Language: En Journal: ACS Med Chem Lett Year: 2010 Document type: Article Country of publication: Estados Unidos