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In vitro, antithrombotic and bleeding time studies of BMS-654457, a small-molecule, reversible and direct inhibitor of factor XIa.
Wong, Pancras C; Quan, Mimi L; Watson, Carol A; Crain, Earl J; Harpel, Mark R; Rendina, Alan R; Luettgen, Joseph M; Wexler, Ruth R; Schumacher, William A; Seiffert, Dietmar A.
Affiliation
  • Wong PC; Cardiovascular Drug Discovery Biology, Bristol-Myers Squibb Company, 311 Pennington-Rocky Hill Road, Pennington, NJ, 08534, USA. pancras.wong@bms.com.
  • Quan ML; Cardiovascular Discovery Chemistry, Bristol-Myers Squibb Company, 311 Pennington-Rocky Hill Road, Pennington, NJ, 08534, USA.
  • Watson CA; Cardiovascular Drug Discovery Biology, Bristol-Myers Squibb Company, 311 Pennington-Rocky Hill Road, Pennington, NJ, 08534, USA.
  • Crain EJ; Cardiovascular Drug Discovery Biology, Bristol-Myers Squibb Company, 311 Pennington-Rocky Hill Road, Pennington, NJ, 08534, USA.
  • Harpel MR; Cardiovascular Drug Discovery Biology, Bristol-Myers Squibb Company, 311 Pennington-Rocky Hill Road, Pennington, NJ, 08534, USA.
  • Rendina AR; Cardiovascular Drug Discovery Biology, Bristol-Myers Squibb Company, 311 Pennington-Rocky Hill Road, Pennington, NJ, 08534, USA.
  • Luettgen JM; Cardiovascular Drug Discovery Biology, Bristol-Myers Squibb Company, 311 Pennington-Rocky Hill Road, Pennington, NJ, 08534, USA.
  • Wexler RR; Cardiovascular Discovery Chemistry, Bristol-Myers Squibb Company, 311 Pennington-Rocky Hill Road, Pennington, NJ, 08534, USA.
  • Schumacher WA; Cardiovascular Drug Discovery Biology, Bristol-Myers Squibb Company, 311 Pennington-Rocky Hill Road, Pennington, NJ, 08534, USA.
  • Seiffert DA; Cardiovascular Drug Discovery Biology, Bristol-Myers Squibb Company, 311 Pennington-Rocky Hill Road, Pennington, NJ, 08534, USA.
J Thromb Thrombolysis ; 40(4): 416-23, 2015 Nov.
Article in En | MEDLINE | ID: mdl-26249722

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Thrombosis / Factor XIa / Fibrinolytic Agents Type of study: Prognostic_studies Limits: Animals / Humans Language: En Journal: J Thromb Thrombolysis Journal subject: ANGIOLOGIA Year: 2015 Document type: Article Affiliation country: Estados Unidos Country of publication: Países Bajos

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Thrombosis / Factor XIa / Fibrinolytic Agents Type of study: Prognostic_studies Limits: Animals / Humans Language: En Journal: J Thromb Thrombolysis Journal subject: ANGIOLOGIA Year: 2015 Document type: Article Affiliation country: Estados Unidos Country of publication: Países Bajos