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JTT-553, a novel Acyl CoA:diacylglycerol acyltransferase (DGAT) 1 inhibitor, improves glucose metabolism in diet-induced obesity and genetic T2DM mice.
Tomimoto, Daisuke; Okuma, Chihiro; Ishii, Yukihito; Kobayashi, Akio; Ohta, Takeshi; Kakutani, Makoto; Imanaka, Tsuneo; Ogawa, Nobuya.
Affiliation
  • Tomimoto D; Central Pharmaceutical Research Institute, Japan Tobacco Inc., 1-1, Murasaki-cho, Takatsuki, Osaka, 569-1125, Japan. Electronic address: daisuke.tomimoto@jt.com.
  • Okuma C; Central Pharmaceutical Research Institute, Japan Tobacco Inc., 1-1, Murasaki-cho, Takatsuki, Osaka, 569-1125, Japan.
  • Ishii Y; Central Pharmaceutical Research Institute, Japan Tobacco Inc., 1-1, Murasaki-cho, Takatsuki, Osaka, 569-1125, Japan.
  • Kobayashi A; Toxicology Research Lab., Central Pharmaceutical Research Institute, Japan Tobacco Inc., 23 Naganuki, Hadano, Kanagawa, 257-0024, Japan.
  • Ohta T; Central Pharmaceutical Research Institute, Japan Tobacco Inc., 1-1, Murasaki-cho, Takatsuki, Osaka, 569-1125, Japan.
  • Kakutani M; Central Pharmaceutical Research Institute, Japan Tobacco Inc., 1-1, Murasaki-cho, Takatsuki, Osaka, 569-1125, Japan.
  • Imanaka T; Cell Biology Laboratory, Graduate School of Medicine and Pharmaceutical Science, University of Toyama, 2630, Sugitani, Toyama-shi, Toyama, 930-0194, Japan.
  • Ogawa N; Central Pharmaceutical Research Institute, Japan Tobacco Inc., 1-1, Murasaki-cho, Takatsuki, Osaka, 569-1125, Japan.
J Pharmacol Sci ; 129(1): 51-8, 2015 Sep.
Article in En | MEDLINE | ID: mdl-26354408

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Oxazines / Spiro Compounds / Body Weight / Weight Gain / Adipose Tissue / Diabetes Mellitus, Type 2 / Diacylglycerol O-Acyltransferase / Glucose / Obesity Type of study: Prognostic_studies Limits: Animals Language: En Journal: J Pharmacol Sci Journal subject: FARMACOLOGIA Year: 2015 Document type: Article

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Oxazines / Spiro Compounds / Body Weight / Weight Gain / Adipose Tissue / Diabetes Mellitus, Type 2 / Diacylglycerol O-Acyltransferase / Glucose / Obesity Type of study: Prognostic_studies Limits: Animals Language: En Journal: J Pharmacol Sci Journal subject: FARMACOLOGIA Year: 2015 Document type: Article