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Structure-Based Discovery of 1H-Indazole-3-carboxamides as a Novel Structural Class of Human GSK-3 Inhibitors.
Ombrato, Rosella; Cazzolla, Nicola; Mancini, Francesca; Mangano, Giorgina.
Affiliation
  • Ombrato R; R&D, Computational Chemistry Laboratory, ‡Chemistry Department, and §In Vitro Pharmacology Development, Angelini Research Center, ACRAF S.p.A. , Piazzale della Stazione, snc, I-00071 Santa Palomba, Pomezia (RM), Italy.
  • Cazzolla N; R&D, Computational Chemistry Laboratory, ‡Chemistry Department, and §In Vitro Pharmacology Development, Angelini Research Center, ACRAF S.p.A. , Piazzale della Stazione, snc, I-00071 Santa Palomba, Pomezia (RM), Italy.
  • Mancini F; R&D, Computational Chemistry Laboratory, ‡Chemistry Department, and §In Vitro Pharmacology Development, Angelini Research Center, ACRAF S.p.A. , Piazzale della Stazione, snc, I-00071 Santa Palomba, Pomezia (RM), Italy.
  • Mangano G; R&D, Computational Chemistry Laboratory, ‡Chemistry Department, and §In Vitro Pharmacology Development, Angelini Research Center, ACRAF S.p.A. , Piazzale della Stazione, snc, I-00071 Santa Palomba, Pomezia (RM), Italy.
J Chem Inf Model ; 55(12): 2540-51, 2015 Dec 28.
Article in En | MEDLINE | ID: mdl-26600430

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Models, Molecular / Dacarbazine / Glycogen Synthase Kinase 3 / Enzyme Inhibitors / Drug Discovery / Indazoles Limits: Humans Language: En Journal: J Chem Inf Model Journal subject: INFORMATICA MEDICA / QUIMICA Year: 2015 Document type: Article Affiliation country: Italia Country of publication: Estados Unidos

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Models, Molecular / Dacarbazine / Glycogen Synthase Kinase 3 / Enzyme Inhibitors / Drug Discovery / Indazoles Limits: Humans Language: En Journal: J Chem Inf Model Journal subject: INFORMATICA MEDICA / QUIMICA Year: 2015 Document type: Article Affiliation country: Italia Country of publication: Estados Unidos