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A Rational Approach for the Identification of Non-Hydroxamate HDAC6-Selective Inhibitors.
Goracci, Laura; Deschamps, Nathalie; Randazzo, Giuseppe Marco; Petit, Charlotte; Dos Santos Passos, Carolina; Carrupt, Pierre-Alain; Simões-Pires, Claudia; Nurisso, Alessandra.
Affiliation
  • Goracci L; School of Pharmaceutical Sciences, University of Geneva, University of Lausanne Quai Ernest-Ansermet, 30, CH-1211, Geneva 4, Switzerland.
  • Deschamps N; Laboratory for Cheminformatics and Molecular Modeling, Department of Chemistry, Biology and Biotechnology, University of Perugia, Via Elce di Sotto, 8, 06123 Perugia, Italy.
  • Randazzo GM; School of Pharmaceutical Sciences, University of Geneva, University of Lausanne Quai Ernest-Ansermet, 30, CH-1211, Geneva 4, Switzerland.
  • Petit C; School of Pharmaceutical Sciences, University of Geneva, University of Lausanne Quai Ernest-Ansermet, 30, CH-1211, Geneva 4, Switzerland.
  • Dos Santos Passos C; School of Pharmaceutical Sciences, University of Geneva, University of Lausanne Quai Ernest-Ansermet, 30, CH-1211, Geneva 4, Switzerland.
  • Carrupt PA; School of Pharmaceutical Sciences, University of Geneva, University of Lausanne Quai Ernest-Ansermet, 30, CH-1211, Geneva 4, Switzerland.
  • Simões-Pires C; School of Pharmaceutical Sciences, University of Geneva, University of Lausanne Quai Ernest-Ansermet, 30, CH-1211, Geneva 4, Switzerland.
  • Nurisso A; School of Pharmaceutical Sciences, University of Geneva, University of Lausanne Quai Ernest-Ansermet, 30, CH-1211, Geneva 4, Switzerland.
Sci Rep ; 6: 29086, 2016 07 12.
Article in En | MEDLINE | ID: mdl-27404291

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Protein Processing, Post-Translational / Histone Deacetylase Inhibitors / Histone Deacetylase 6 / Neoplasms Type of study: Diagnostic_studies Limits: Humans Language: En Journal: Sci Rep Year: 2016 Document type: Article Affiliation country: Suiza

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Protein Processing, Post-Translational / Histone Deacetylase Inhibitors / Histone Deacetylase 6 / Neoplasms Type of study: Diagnostic_studies Limits: Humans Language: En Journal: Sci Rep Year: 2016 Document type: Article Affiliation country: Suiza