Discovery of Tropifexor (LJN452), a Highly Potent Non-bile Acid FXR Agonist for the Treatment of Cholestatic Liver Diseases and Nonalcoholic Steatohepatitis (NASH).
J Med Chem
; 60(24): 9960-9973, 2017 12 28.
Article
in En
| MEDLINE
| ID: mdl-29148806
Full text:
1
Collection:
01-internacional
Database:
MEDLINE
Main subject:
Cholestasis
/
Receptors, Cytoplasmic and Nuclear
/
Benzothiazoles
/
Non-alcoholic Fatty Liver Disease
/
Isoxazoles
Type of study:
Prognostic_studies
Limits:
Animals
/
Humans
/
Male
Language:
En
Journal:
J Med Chem
Journal subject:
QUIMICA
Year:
2017
Document type:
Article
Affiliation country:
Estados Unidos