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Structure-based design and discovery of potent and selective KDM5 inhibitors.
Nie, Zhe; Shi, Lihong; Lai, Chon; O'Connell, Shawn M; Xu, Jiangchun; Stansfield, Ryan K; Hosfield, David J; Veal, James M; Stafford, Jeffrey A.
Affiliation
  • Nie Z; Celgene Corporation, 10300 Campus Point Drive, Suite 100, San Diego, CA 92121, USA. Electronic address: znie@celgene.com.
  • Shi L; Celgene Corporation, 10300 Campus Point Drive, Suite 100, San Diego, CA 92121, USA.
  • Lai C; Celgene Corporation, 10300 Campus Point Drive, Suite 100, San Diego, CA 92121, USA.
  • O'Connell SM; Celgene Corporation, 10300 Campus Point Drive, Suite 100, San Diego, CA 92121, USA.
  • Xu J; Celgene Corporation, 10300 Campus Point Drive, Suite 100, San Diego, CA 92121, USA.
  • Stansfield RK; Celgene Corporation, 10300 Campus Point Drive, Suite 100, San Diego, CA 92121, USA.
  • Hosfield DJ; Ben May Department for Cancer Research, University of Chicago, 929 East 57th Street, Chicago, IL 60637, USA.
  • Veal JM; Celgene Corporation, 10300 Campus Point Drive, Suite 100, San Diego, CA 92121, USA.
  • Stafford JA; Celgene Corporation, 10300 Campus Point Drive, Suite 100, San Diego, CA 92121, USA.
Bioorg Med Chem Lett ; 28(9): 1490-1494, 2018 05 15.
Article in En | MEDLINE | ID: mdl-29627262
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Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Repressor Proteins / Nuclear Proteins / Enzyme Inhibitors / Drug Discovery / Jumonji Domain-Containing Histone Demethylases / Retinoblastoma-Binding Protein 2 / Antineoplastic Agents Type of study: Prognostic_studies Limits: Female / Humans Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2018 Document type: Article
Fulltext
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Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Repressor Proteins / Nuclear Proteins / Enzyme Inhibitors / Drug Discovery / Jumonji Domain-Containing Histone Demethylases / Retinoblastoma-Binding Protein 2 / Antineoplastic Agents Type of study: Prognostic_studies Limits: Female / Humans Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2018 Document type: Article