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Design, Synthesis, and Testing of Potent, Selective Hepsin Inhibitors via Application of an Automated Closed-Loop Optimization Platform.
Pant, Shishir M; Mukonoweshuro, Amanda; Desai, Bimbisar; Ramjee, Manoj K; Selway, Christopher N; Tarver, Gary J; Wright, Adrian G; Birchall, Kristian; Chapman, Timothy M; Tervonen, Topi A; Klefström, Juha.
Affiliation
  • Pant SM; Cancer Cell Circuitry Laboratory, Research Programs Unit/Translational Cancer Biology & Medicum, University of Helsinki , P.O. Box 63, Haartmaninkatu 8 , 00014 Helsinki , Finland.
  • Mukonoweshuro A; Cyclofluidic Ltd. , Biopark, Broadwater Road , Welwyn Garden City , AL7 3AX , U.K.
  • Desai B; Cyclofluidic Ltd. , Biopark, Broadwater Road , Welwyn Garden City , AL7 3AX , U.K.
  • Ramjee MK; Cyclofluidic Ltd. , Biopark, Broadwater Road , Welwyn Garden City , AL7 3AX , U.K.
  • Selway CN; Cyclofluidic Ltd. , Biopark, Broadwater Road , Welwyn Garden City , AL7 3AX , U.K.
  • Tarver GJ; Cyclofluidic Ltd. , Biopark, Broadwater Road , Welwyn Garden City , AL7 3AX , U.K.
  • Wright AG; Cyclofluidic Ltd. , Biopark, Broadwater Road , Welwyn Garden City , AL7 3AX , U.K.
  • Birchall K; LifeArc , Accelerator Building, Open Innovation Campus , Stevenage , SG1 2FX , U.K.
  • Chapman TM; LifeArc , Accelerator Building, Open Innovation Campus , Stevenage , SG1 2FX , U.K.
  • Tervonen TA; Cancer Cell Circuitry Laboratory, Research Programs Unit/Translational Cancer Biology & Medicum, University of Helsinki , P.O. Box 63, Haartmaninkatu 8 , 00014 Helsinki , Finland.
  • Klefström J; Cancer Cell Circuitry Laboratory, Research Programs Unit/Translational Cancer Biology & Medicum, University of Helsinki , P.O. Box 63, Haartmaninkatu 8 , 00014 Helsinki , Finland.
J Med Chem ; 61(10): 4335-4347, 2018 05 24.
Article in En | MEDLINE | ID: mdl-29701962

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Breast Neoplasms / Serine Endopeptidases / Drug Design / Cell Proliferation / Enzyme Inhibitors / High-Throughput Screening Assays Type of study: Prognostic_studies Limits: Female / Humans Language: En Journal: J Med Chem Journal subject: QUIMICA Year: 2018 Document type: Article Affiliation country: Finlandia Country of publication: Estados Unidos

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Breast Neoplasms / Serine Endopeptidases / Drug Design / Cell Proliferation / Enzyme Inhibitors / High-Throughput Screening Assays Type of study: Prognostic_studies Limits: Female / Humans Language: En Journal: J Med Chem Journal subject: QUIMICA Year: 2018 Document type: Article Affiliation country: Finlandia Country of publication: Estados Unidos