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In vitro and in vivo metabolic investigation of the Palbociclib by UHPLC-Q-TOF/MS/MS and in silico toxicity studies of its metabolites.
Chavan, Balasaheb B; Tiwari, Shristy; G, Shankar; Nimbalkar, Rakesh D; Garg, Prabha; R, Srinivas; Talluri, M V N Kumar.
Affiliation
  • Chavan BB; Department of Pharmaceutical Analysis, National Institute of Pharmaceutical Education & Research, IDPL R&D Campus, Balanagar, Hyderabad, 500 037, India.
  • Tiwari S; Department of Pharmaceutical Analysis, National Institute of Pharmaceutical Education & Research, IDPL R&D Campus, Balanagar, Hyderabad, 500 037, India.
  • G S; National Center for Mass Spectrometry, CSIR-Indian Institute of Chemical Technology, Tarnaka, Hyderabad, 500 607, India.
  • Nimbalkar RD; National Institute of Pharmaceutical Education and Research (NIPER), Sector 67, S.A.S. Nagar, 160 062, Punjab, India.
  • Garg P; National Institute of Pharmaceutical Education and Research (NIPER), Sector 67, S.A.S. Nagar, 160 062, Punjab, India.
  • R S; Department of Pharmaceutical Analysis, National Institute of Pharmaceutical Education & Research, IDPL R&D Campus, Balanagar, Hyderabad, 500 037, India; National Center for Mass Spectrometry, CSIR-Indian Institute of Chemical Technology, Tarnaka, Hyderabad, 500 607, India.
  • Talluri MVNK; Department of Pharmaceutical Analysis, National Institute of Pharmaceutical Education & Research, IDPL R&D Campus, Balanagar, Hyderabad, 500 037, India. Electronic address: narendra@niperhyd.ac.in.
J Pharm Biomed Anal ; 157: 59-74, 2018 Aug 05.
Article in En | MEDLINE | ID: mdl-29772457

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Piperazines / Pyridines Limits: Animals / Humans / Male Language: En Journal: J Pharm Biomed Anal Year: 2018 Document type: Article Affiliation country: India Country of publication: Reino Unido

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Piperazines / Pyridines Limits: Animals / Humans / Male Language: En Journal: J Pharm Biomed Anal Year: 2018 Document type: Article Affiliation country: India Country of publication: Reino Unido