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Impact of Ethnicity-Specific Hepatic Microsomal Scaling Factor, Liver Weight, and Cytochrome P450 (CYP) 1A2 Content on Physiologically Based Prediction of CYP1A2-Mediated Pharmacokinetics in Young and Elderly Chinese Adults.
Li, Guo-Fu; Zheng, Qing-Shan; Yu, Yichao; Zhong, Wei; Zhou, Hong-Hao; Qiu, Furong; Wang, Guangji; Yu, Guo; Derendorf, Hartmut.
Affiliation
  • Li GF; Clinical Medical College, Yangzhou University, #98 West Nantong Rd., Yangzhou, Jiangsu, China.
  • Zheng QS; Department of Pharmaceutics, College of Pharmacy, University of Florida, 1345 Center Drive, P3-27, Gainesville, FL, 32610-0494, USA.
  • Yu Y; Center for Drug Clinical Research, Shanghai University of Chinese Medicine, Shanghai, China.
  • Zhong W; Center for Drug Clinical Research, Shanghai University of Chinese Medicine, Shanghai, China.
  • Zhou HH; Department of Pharmaceutics, College of Pharmacy, University of Florida, 1345 Center Drive, P3-27, Gainesville, FL, 32610-0494, USA.
  • Qiu F; Clinical Medical College, Yangzhou University, #98 West Nantong Rd., Yangzhou, Jiangsu, China.
  • Wang G; Department of Clinical Pharmacology, Xiangya Hospital, Central South University, Changsha, Hunan, China.
  • Yu G; Laboratory of Clinical Pharmacokinetics, Shuguang Hospital, Shanghai University of Chinese Medicine, Shanghai, China.
  • Derendorf H; Key Lab of Drug Metabolism and Pharmacokinetics, China, Pharmaceutical University, Nanjing, Jiangsu, China.
Clin Pharmacokinet ; 58(7): 927-941, 2019 07.
Article in En | MEDLINE | ID: mdl-30767128

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Microsomes, Liver / Cytochrome P-450 CYP1A2 / Liver / Models, Biological Type of study: Prognostic_studies / Risk_factors_studies Aspects: Determinantes_sociais_saude Limits: Adult / Aged / Female / Humans / Male / Middle aged Language: En Journal: Clin Pharmacokinet Year: 2019 Document type: Article Affiliation country: China Country of publication: Suiza

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Microsomes, Liver / Cytochrome P-450 CYP1A2 / Liver / Models, Biological Type of study: Prognostic_studies / Risk_factors_studies Aspects: Determinantes_sociais_saude Limits: Adult / Aged / Female / Humans / Male / Middle aged Language: En Journal: Clin Pharmacokinet Year: 2019 Document type: Article Affiliation country: China Country of publication: Suiza