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Lack of a Clinically Significant Pharmacokinetic Interaction between Etravirine and Raltegravir Using an Original Approach Based on Drug Metabolism, Protein Binding, and Penetration in Seminal Fluid: A Pharmacokinetic Substudy of the ANRS-163 ETRAL Study.
Lê, Minh Patrick; Valantin, Marc-Antoine; Assoumou, Lambert; Soulie, Cathia; Le Mestre, Soizic; Weiss, Laurence; Yazdanpanah, Yazdan; Molina, Jean-Michel; Bouchaud, Olivier; Raffi, François; Reynes, Jacques; Calvez, Vincent; Marcelin, Anne-Geneviève; Costagliola, Dominique; Katlama, Christine; Peytavin, Gilles.
Affiliation
  • Lê MP; IAME, UMR 1137, Sorbonne Paris Cité and INSERM, Université Paris Diderot, Paris, France.
  • Valantin MA; Laboratoire de Pharmacologie-Toxicologie, AP-HP, Hôpital Bichat-Claude Bernard, Paris, France.
  • Assoumou L; Service de Maladies Infectieuses et Tropicales, AP-HP, Hôpital Pitié-Salpêtrière, Paris, France.
  • Soulie C; INSERM, Institut Pierre Louis d'Epidémiologie et de Santé Publique (iPLESP UMRS 1136), Sorbonne Université, UPMC Univ Paris 06, Paris, France.
  • Le Mestre S; INSERM, Institut Pierre Louis d'Epidémiologie et de Santé Publique (iPLESP UMRS 1136), Sorbonne Université, UPMC Univ Paris 06, Paris, France.
  • Weiss L; Laboratoire de Virologie, INSERM, Institut Pierre Louis d'Epidémiologie et de Santé Publique (iPLESP), AP-HP, Hôpital Pitié Salpêtrière, Sorbonne Université, Paris, France.
  • Yazdanpanah Y; France Recherche Nord & Sud SIDA-HIV Hépatites (ANRS), Paris, France.
  • Molina JM; Service d'Immunologie Clinique, AP-HP, Hôpital Européen Georges Pompidou, Paris, France.
  • Bouchaud O; IAME, UMR 1137, Sorbonne Paris Cité and INSERM, Université Paris Diderot, Paris, France.
  • Raffi F; Service de Maladies Infectieuses et Tropicales, AP-HP, Hôpital Bichat-Claude Bernard, Paris, France.
  • Reynes J; Service de Maladies Infectieuses et Tropicales, INSERM U941, AP-HP, Hôpital Saint Louis, Université Denis Diderot Paris VII, Paris, France.
  • Calvez V; Service de Maladies Infectieuses et Tropicales, AP-HP, Hôpital Avicenne, Bobigny, France.
  • Marcelin AG; Department of Infectious Diseases, Hotel-Dieu Hospital - INSERM CIC 1413, Nantes University Hospital, Nantes, France.
  • Costagliola D; Service de Maladies Infectieuses et Tropicales, CHU Montpellier, Montpellier, France.
  • Katlama C; INSERM U1175, IRD UMI 233, University of Montpellier, Montpellier, France.
  • Peytavin G; Laboratoire de Virologie, INSERM, Institut Pierre Louis d'Epidémiologie et de Santé Publique (iPLESP), AP-HP, Hôpital Pitié Salpêtrière, Sorbonne Université, Paris, France.
Pharmacotherapy ; 39(4): 514-520, 2019 04.
Article in En | MEDLINE | ID: mdl-30815916

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Pyridazines / Semen / HIV Infections / Anti-HIV Agents / Raltegravir Potassium Limits: Female / Humans / Male / Middle aged Language: En Journal: Pharmacotherapy Year: 2019 Document type: Article Affiliation country: Francia

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Pyridazines / Semen / HIV Infections / Anti-HIV Agents / Raltegravir Potassium Limits: Female / Humans / Male / Middle aged Language: En Journal: Pharmacotherapy Year: 2019 Document type: Article Affiliation country: Francia