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Pharmacology of JNJ-28583113: A novel TRPM2 antagonist.
Fourgeaud, Lawrence; Dvorak, Curt; Faouzi, Malika; Starkus, John; Sahdeo, Sunil; Wang, Qi; Lord, Brian; Coate, Heather; Taylor, Natalie; He, Yingbo; Qin, Ning; Wickenden, Alan; Carruthers, Nicholas; Lovenberg, Timothy W; Penner, Reinhold; Bhattacharya, Anindya.
Affiliation
  • Fourgeaud L; Janssen Research & Development, LLC, 3210 Merryfield Row, San Diego, CA, 92121, USA. Electronic address: lfourgea@its.jnj.com.
  • Dvorak C; Janssen Research & Development, LLC, 3210 Merryfield Row, San Diego, CA, 92121, USA.
  • Faouzi M; Centre for Biomedical Research at the Queen's Medical Centre, Honolulu, HI, 96813, USA.
  • Starkus J; Centre for Biomedical Research at the Queen's Medical Centre, Honolulu, HI, 96813, USA.
  • Sahdeo S; Janssen Research & Development, LLC, 3210 Merryfield Row, San Diego, CA, 92121, USA.
  • Wang Q; Janssen Research & Development, LLC, 3210 Merryfield Row, San Diego, CA, 92121, USA.
  • Lord B; Janssen Research & Development, LLC, 3210 Merryfield Row, San Diego, CA, 92121, USA.
  • Coate H; Janssen Research & Development, LLC, 3210 Merryfield Row, San Diego, CA, 92121, USA.
  • Taylor N; Janssen Research & Development, LLC, 3210 Merryfield Row, San Diego, CA, 92121, USA.
  • He Y; Janssen Research & Development, LLC, 3210 Merryfield Row, San Diego, CA, 92121, USA.
  • Qin N; Janssen Research & Development, LLC, 3210 Merryfield Row, San Diego, CA, 92121, USA.
  • Wickenden A; Janssen Research & Development, LLC, 3210 Merryfield Row, San Diego, CA, 92121, USA.
  • Carruthers N; Janssen Research & Development, LLC, 3210 Merryfield Row, San Diego, CA, 92121, USA.
  • Lovenberg TW; Janssen Research & Development, LLC, 3210 Merryfield Row, San Diego, CA, 92121, USA.
  • Penner R; Centre for Biomedical Research at the Queen's Medical Centre, Honolulu, HI, 96813, USA.
  • Bhattacharya A; Janssen Research & Development, LLC, 3210 Merryfield Row, San Diego, CA, 92121, USA.
Eur J Pharmacol ; 853: 299-307, 2019 Jun 15.
Article in En | MEDLINE | ID: mdl-30965058

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Pyrazoles / TRPM Cation Channels / Drug Discovery Limits: Animals / Humans / Male Language: En Journal: Eur J Pharmacol Year: 2019 Document type: Article Country of publication: Países Bajos

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Pyrazoles / TRPM Cation Channels / Drug Discovery Limits: Animals / Humans / Male Language: En Journal: Eur J Pharmacol Year: 2019 Document type: Article Country of publication: Países Bajos