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Optimization of 4-Aminopiperidines as Inhibitors of Influenza A Viral Entry That Are Synergistic with Oseltamivir.
Gaisina, Irina N; Peet, Norton P; Cheng, Han; Li, Ping; Du, Ruikun; Cui, Qinghua; Furlong, Kevin; Manicassamy, Balaji; Caffrey, Michael; Thatcher, Gregory R J; Rong, Lijun.
Affiliation
  • Gaisina IN; UICentre (Drug Discovery@UIC) and Department of Pharmaceutical Sciences, College of Pharmacy, University of Illinois at Chicago, 833 South Wood Street, Chicago, Illinois 60612, United States.
  • Peet NP; Chicago BioSolutions, Inc., 2242 West Harrison Street, Chicago, Illinois 60612, United States.
  • Cheng H; Chicago BioSolutions, Inc., 2242 West Harrison Street, Chicago, Illinois 60612, United States.
  • Li P; Department of Microbiology and Immunology, College of Medicine, University of Illinois at Chicago, 909 South Wolcott Avenue, Chicago, Illinois 60612, United States.
  • Du R; College of Pharmacy, Shandong University of Traditional Chinese Medicine, 16369 Jinshi Road, Jinan, Shandong 250355, China.
  • Cui Q; College of Pharmacy, Shandong University of Traditional Chinese Medicine, 16369 Jinshi Road, Jinan, Shandong 250355, China.
  • Furlong K; College of Pharmacy, Shandong University of Traditional Chinese Medicine, 16369 Jinshi Road, Jinan, Shandong 250355, China.
  • Manicassamy B; Department of Microbiology, University of Chicago, 920 East 58th Street, Chicago, Illinois 60637, United States.
  • Caffrey M; Department of Microbiology, University of Chicago, 920 East 58th Street, Chicago, Illinois 60637, United States.
  • Thatcher GRJ; Department of Microbiology and Immunology, University of Iowa, 51 Newton Road, Iowa City, Iowa 52242, United States.
  • Rong L; Department of Biochemistry and Molecular Genetics, College of Medicine, University of Illinois at Chicago, 900 South Ashland Avenue, Chicago, Illinois 60607, United States.
J Med Chem ; 63(6): 3120-3130, 2020 03 26.
Article in En | MEDLINE | ID: mdl-32069052

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Antiviral Agents / Piperidines / Influenza A Virus, H1N1 Subtype / Influenza A Virus, H5N1 Subtype / Oseltamivir / Virus Internalization Limits: Animals / Humans Language: En Journal: J Med Chem Journal subject: QUIMICA Year: 2020 Document type: Article Affiliation country: Estados Unidos Country of publication: Estados Unidos

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Antiviral Agents / Piperidines / Influenza A Virus, H1N1 Subtype / Influenza A Virus, H5N1 Subtype / Oseltamivir / Virus Internalization Limits: Animals / Humans Language: En Journal: J Med Chem Journal subject: QUIMICA Year: 2020 Document type: Article Affiliation country: Estados Unidos Country of publication: Estados Unidos