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Early Drug-Discovery Efforts towards the Identification of EP300/CBP Histone Acetyltransferase (HAT) Inhibitors.
Huhn, Annissa J; Gardberg, Anna S; Poy, Florence; Brucelle, Francois; Vivat, Valerie; Cantone, Nico; Patel, Gaurav; Patel, Chirag; Cummings, Richard; Sims, Robert; Levell, Julian; Audia, James E; Bommi-Reddy, Archana; Wilson, Jonathan E.
Affiliation
  • Huhn AJ; Constellation Pharmaceuticals, 215 First Street, Cambridge, MA 02142.
  • Gardberg AS; Constellation Pharmaceuticals, 215 First Street, Cambridge, MA 02142.
  • Poy F; Constellation Pharmaceuticals, 215 First Street, Cambridge, MA 02142.
  • Brucelle F; Foghorn Therapeutics, 100 Binney St., Cambridge, MA 02142.
  • Vivat V; Constellation Pharmaceuticals, 215 First Street, Cambridge, MA 02142.
  • Cantone N; Constellation Pharmaceuticals, 215 First Street, Cambridge, MA 02142.
  • Patel G; Piramal Enterprises Limited-Discovery Solutions Ahmedabad, Gujarat, 382 213.
  • Patel C; Piramal Enterprises Limited-Discovery Solutions Ahmedabad, Gujarat, 382 213.
  • Cummings R; Constellation Pharmaceuticals, 215 First Street, Cambridge, MA 02142.
  • Sims R; Third Rock Ventures, 29 Newbury St. #301, Boston, MA 02116.
  • Levell J; Constellation Pharmaceuticals, 215 First Street, Cambridge, MA 02142.
  • Audia JE; Third Rock Ventures, 29 Newbury St. #301, Boston, MA 02116.
  • Bommi-Reddy A; Constellation Pharmaceuticals, 215 First Street, Cambridge, MA 02142.
  • Wilson JE; Constellation Pharmaceuticals, 215 First Street, Cambridge, MA 02142.
ChemMedChem ; 15(11): 955-960, 2020 06 04.
Article in En | MEDLINE | ID: mdl-32181984

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Enzyme Inhibitors / P300-CBP Transcription Factors / Drug Discovery Type of study: Diagnostic_studies / Prognostic_studies Limits: Humans Language: En Journal: ChemMedChem Journal subject: FARMACOLOGIA / QUIMICA Year: 2020 Document type: Article Country of publication: Alemania

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Enzyme Inhibitors / P300-CBP Transcription Factors / Drug Discovery Type of study: Diagnostic_studies / Prognostic_studies Limits: Humans Language: En Journal: ChemMedChem Journal subject: FARMACOLOGIA / QUIMICA Year: 2020 Document type: Article Country of publication: Alemania