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New insights on the arylpiperazinylalkyl pyridazinone ET1 as potent antinociceptive and anti-inflammatory agent.
Μaione, Francesco; Colucci, Mariantonella; Raucci, Federica; Mangano, Giorgina; Marzoli, Francesca; Mascolo, Nicola; Crocetti, Letizia; Giovannoni, Maria Paola; Di Giannuario, Amalia; Pieretti, Stefano.
Affiliation
  • Μaione F; ImmunoPharmaLab, Department of Pharmacy, School of Medicine and Surgery, University of Naples Federico II, Via Domenico Montesano 49, 80131, Naples, Italy.
  • Colucci M; National Center for Drug Research and Evaluation, Istituto Superiore di Sanità, Viale Regina Elena 299, 00161, Rome, Italy.
  • Raucci F; ImmunoPharmaLab, Department of Pharmacy, School of Medicine and Surgery, University of Naples Federico II, Via Domenico Montesano 49, 80131, Naples, Italy.
  • Mangano G; Angelini RR&D (Regulatory, Research & Development), Angelini Pharma S.p.A., Piazzale della Stazione SNC, S. Palomba-Pomezia, Rome, 00071, Italy.
  • Marzoli F; National Center for Drug Research and Evaluation, Istituto Superiore di Sanità, Viale Regina Elena 299, 00161, Rome, Italy.
  • Mascolo N; ImmunoPharmaLab, Department of Pharmacy, School of Medicine and Surgery, University of Naples Federico II, Via Domenico Montesano 49, 80131, Naples, Italy.
  • Crocetti L; NEUROFARBA, Pharmaceutical and Nutraceutical Section, University of Florence, 50019, Sesto Fiorentino, Italy.
  • Giovannoni MP; NEUROFARBA, Pharmaceutical and Nutraceutical Section, University of Florence, 50019, Sesto Fiorentino, Italy.
  • Di Giannuario A; National Center for Drug Research and Evaluation, Istituto Superiore di Sanità, Viale Regina Elena 299, 00161, Rome, Italy.
  • Pieretti S; National Center for Drug Research and Evaluation, Istituto Superiore di Sanità, Viale Regina Elena 299, 00161, Rome, Italy. Electronic address: stefano.pieretti@iss.it.
Eur J Pharmacol ; 888: 173572, 2020 Dec 05.
Article in En | MEDLINE | ID: mdl-32946866

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Pain / Pyridazines / Pain Measurement / Analgesics / Anti-Inflammatory Agents Limits: Animals / Humans / Male Language: En Journal: Eur J Pharmacol Year: 2020 Document type: Article Affiliation country: Italia Country of publication: Países Bajos

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Pain / Pyridazines / Pain Measurement / Analgesics / Anti-Inflammatory Agents Limits: Animals / Humans / Male Language: En Journal: Eur J Pharmacol Year: 2020 Document type: Article Affiliation country: Italia Country of publication: Países Bajos