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An innovative kinome platform to accelerate small-molecule inhibitor discovery and optimization from hits to leads.
Chaudhry, Charu; Tebben, Andrew; Tokarski, John S; Borzilleri, Robert; Pitts, William J; Lippy, Jonathan; Zhang, Litao.
Affiliation
  • Chaudhry C; Lead Discovery and Optimization, Bristol Myers Squibb, NJ, USA. Electronic address: cchaudhr@its.jnj.com.
  • Tebben A; Molecular Structure and Design, Molecular Discovery Technologies, Bristol Myers Squibb, NJ, USA.
  • Tokarski JS; Molecular Structure and Design, Molecular Discovery Technologies, Bristol Myers Squibb, NJ, USA.
  • Borzilleri R; Oncology Discovery Chemistry, Bristol Myers Squibb, NJ, USA.
  • Pitts WJ; Immunosciences Discovery Chemistry, Bristol Myers Squibb, NJ, USA.
  • Lippy J; Lead Discovery and Optimization, Bristol Myers Squibb, NJ, USA.
  • Zhang L; Lead Discovery and Optimization, Bristol Myers Squibb, NJ, USA.
Drug Discov Today ; 26(5): 1115-1125, 2021 05.
Article in En | MEDLINE | ID: mdl-33497831

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Protein Kinases / Protein Kinase Inhibitors / Drug Discovery Limits: Animals / Humans Country/Region as subject: America do norte Language: En Journal: Drug Discov Today Journal subject: FARMACOLOGIA / TERAPIA POR MEDICAMENTOS Year: 2021 Document type: Article Country of publication: Reino Unido

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Protein Kinases / Protein Kinase Inhibitors / Drug Discovery Limits: Animals / Humans Country/Region as subject: America do norte Language: En Journal: Drug Discov Today Journal subject: FARMACOLOGIA / TERAPIA POR MEDICAMENTOS Year: 2021 Document type: Article Country of publication: Reino Unido