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CLIPSing Melanotan-II to Discover Multiple Functionally Selective hMCR Agonists.
Tomassi, Stefano; Dimmito, Marilisa Pia; Cai, Minying; D'Aniello, Antonia; Del Bene, Alessandra; Messere, Anna; Liu, Zekun; Zhu, Tingyi; Hruby, Victor J; Stefanucci, Azzurra; Cosconati, Sandro; Mollica, Adriano; Di Maro, Salvatore.
Affiliation
  • Tomassi S; Dipartimento di Farmacia, Università degli Studi di Napoli "Federico II", Via D. Montesano 49, Naples 80131, Italy.
  • Dimmito MP; Dipartimento di Farmacia, Università di Chieti-Pescara "G. d'Annunzio", Via dei Vestini 31, Chieti 66100, Italy.
  • Cai M; Department of Chemistry and Biochemistry, University of Arizona, Tucson, Arizona 85721, United States.
  • D'Aniello A; DiSTABiF, University of Campania "Luigi Vanvitelli", Via Vivaldi 43, 81100 Caserta, Italy.
  • Del Bene A; DiSTABiF, University of Campania "Luigi Vanvitelli", Via Vivaldi 43, 81100 Caserta, Italy.
  • Messere A; DiSTABiF, University of Campania "Luigi Vanvitelli", Via Vivaldi 43, 81100 Caserta, Italy.
  • Liu Z; Department of Chemistry and Biochemistry, University of Arizona, Tucson, Arizona 85721, United States.
  • Zhu T; Department of Chemistry and Biochemistry, University of Arizona, Tucson, Arizona 85721, United States.
  • Hruby VJ; Department of Chemistry and Biochemistry, University of Arizona, Tucson, Arizona 85721, United States.
  • Stefanucci A; Dipartimento di Farmacia, Università di Chieti-Pescara "G. d'Annunzio", Via dei Vestini 31, Chieti 66100, Italy.
  • Cosconati S; DiSTABiF, University of Campania "Luigi Vanvitelli", Via Vivaldi 43, 81100 Caserta, Italy.
  • Mollica A; Dipartimento di Farmacia, Università di Chieti-Pescara "G. d'Annunzio", Via dei Vestini 31, Chieti 66100, Italy.
  • Di Maro S; DiSTABiF, University of Campania "Luigi Vanvitelli", Via Vivaldi 43, 81100 Caserta, Italy.
J Med Chem ; 65(5): 4007-4017, 2022 03 10.
Article in En | MEDLINE | ID: mdl-35188390

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Alpha-MSH / Receptors, Melanocortin Limits: Humans Language: En Journal: J Med Chem Journal subject: QUIMICA Year: 2022 Document type: Article Affiliation country: Italia

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Alpha-MSH / Receptors, Melanocortin Limits: Humans Language: En Journal: J Med Chem Journal subject: QUIMICA Year: 2022 Document type: Article Affiliation country: Italia