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Small molecule peptidomimetic trypsin inhibitors: validation of an EKO binding mode, but with a twist.
Lyu, Rui-Liang; Joy, Shaon; Packianathan, Charles; Laganowsky, Arthur; Burgess, Kevin.
Affiliation
  • Lyu RL; Department of Chemistry, Texas A & M University, Box 30012, College Station, TX 77842-3012, USA. burgess@tamu.edu.
  • Joy S; Department of Chemistry, Texas A & M University, Box 30012, College Station, TX 77842-3012, USA. burgess@tamu.edu.
  • Packianathan C; Department of Chemistry, Texas A & M University, Box 30012, College Station, TX 77842-3012, USA. burgess@tamu.edu.
  • Laganowsky A; Department of Chemistry, Texas A & M University, Box 30012, College Station, TX 77842-3012, USA. burgess@tamu.edu.
  • Burgess K; Department of Chemistry, Texas A & M University, Box 30012, College Station, TX 77842-3012, USA. burgess@tamu.edu.
Org Biomol Chem ; 20(10): 2075-2080, 2022 03 09.
Article in En | MEDLINE | ID: mdl-35225309
Subject(s)

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Trypsin Inhibitors Language: En Journal: Org Biomol Chem Journal subject: BIOQUIMICA / QUIMICA Year: 2022 Document type: Article Affiliation country: Estados Unidos Country of publication: Reino Unido

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Trypsin Inhibitors Language: En Journal: Org Biomol Chem Journal subject: BIOQUIMICA / QUIMICA Year: 2022 Document type: Article Affiliation country: Estados Unidos Country of publication: Reino Unido