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Design, synthesis and biological evaluation of novel 9-methyl-9H-purine and thieno[3, 2-d]pyrimidine derivatives as potent mTOR inhibitors.
Yang, Ying-Yue; Wang, Wan-Li; Hu, Xia-Tong; Chen, Xin; Ni, Yang; Lei, Yan-Hua; Qiu, Qi-Yuan; Tao, Long-Yue; Luo, Tian-Wen; Wang, Ning-Yu.
Affiliation
  • Yang YY; School of Life Science and Engineering, Southwest Jiaotong University, Chengdu, China.
  • Wang WL; School of Life Science and Engineering, Southwest Jiaotong University, Chengdu, China.
  • Hu XT; School of Life Science and Engineering, Southwest Jiaotong University, Chengdu, China.
  • Chen X; School of Life Science and Engineering, Southwest Jiaotong University, Chengdu, China.
  • Ni Y; School of Life Science and Engineering, Southwest Jiaotong University, Chengdu, China.
  • Lei YH; School of Life Science and Engineering, Southwest Jiaotong University, Chengdu, China.
  • Qiu QY; School of Life Science and Engineering, Southwest Jiaotong University, Chengdu, China.
  • Tao LY; State Key Laboratory of Biotherapy and Cancer Center, West China Hospital, and Collaborative Innovation Center of Biotherapy, Sichuan University, Chengdu, China.
  • Luo TW; State Key Laboratory of Biotherapy and Cancer Center, West China Hospital, and Collaborative Innovation Center of Biotherapy, Sichuan University, Chengdu, China.
  • Wang NY; School of Life Science and Engineering, Southwest Jiaotong University, Chengdu, China. Electronic address: wangny-swjtu@swjtu.edu.cn.
Bioorg Chem ; 132: 106356, 2023 03.
Article in En | MEDLINE | ID: mdl-36669357

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Neoplasms / Antineoplastic Agents Limits: Humans Language: En Journal: Bioorg Chem Year: 2023 Document type: Article Affiliation country: China Country of publication: Estados Unidos

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Neoplasms / Antineoplastic Agents Limits: Humans Language: En Journal: Bioorg Chem Year: 2023 Document type: Article Affiliation country: China Country of publication: Estados Unidos