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Rapid optimisation of fragments and hits to lead compounds from screening of crude reaction mixtures.
Baker, Lisa M; Aimon, Anthony; Murray, James B; Surgenor, Allan E; Matassova, Natalia; Roughley, Stephen D; Collins, Patrick M; Krojer, Tobias; von Delft, Frank; Hubbard, Roderick E.
Affiliation
  • Baker LM; Vernalis (R&D) Ltd, Granta Park, Cambridge, CB21 6GB, UK.
  • Aimon A; Diamond Light Source Ltd., Harwell Science and Innovation Campus, Didcot, OX11 0QX, UK.
  • Murray JB; Research Complex at Harwell (RCaH), Rutherford Appleton Laboratory, Didcot, OX11 0FA, UK.
  • Surgenor AE; Vernalis (R&D) Ltd, Granta Park, Cambridge, CB21 6GB, UK.
  • Matassova N; Vernalis (R&D) Ltd, Granta Park, Cambridge, CB21 6GB, UK.
  • Roughley SD; Vernalis (R&D) Ltd, Granta Park, Cambridge, CB21 6GB, UK.
  • Collins PM; Vernalis (R&D) Ltd, Granta Park, Cambridge, CB21 6GB, UK.
  • Krojer T; Diamond Light Source Ltd., Harwell Science and Innovation Campus, Didcot, OX11 0QX, UK.
  • von Delft F; Structural Genomics Consortium (SGC), University of Oxford, Oxford, OX3 7DQ, UK.
  • Hubbard RE; Diamond Light Source Ltd., Harwell Science and Innovation Campus, Didcot, OX11 0QX, UK.
Commun Chem ; 3(1): 122, 2020 Sep 02.
Article in En | MEDLINE | ID: mdl-36703375

Full text: 1 Collection: 01-internacional Database: MEDLINE Type of study: Diagnostic_studies / Screening_studies Language: En Journal: Commun Chem Year: 2020 Document type: Article Affiliation country: Reino Unido Country of publication: Reino Unido

Full text: 1 Collection: 01-internacional Database: MEDLINE Type of study: Diagnostic_studies / Screening_studies Language: En Journal: Commun Chem Year: 2020 Document type: Article Affiliation country: Reino Unido Country of publication: Reino Unido