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Discovery and Characterization of BAY-805, a Potent and Selective Inhibitor of Ubiquitin-Specific Protease USP21.
Göricke, Fabian; Vu, Victoria; Smith, Leanna; Scheib, Ulrike; Böhm, Raphael; Akkilic, Namik; Wohlfahrt, Gerd; Weiske, Jörg; Bömer, Ulf; Brzezinka, Krzysztof; Lindner, Niels; Lienau, Philip; Gradl, Stefan; Beck, Hartmut; Brown, Peter J; Santhakumar, Vijayaratnam; Vedadi, Masoud; Barsyte-Lovejoy, Dalia; Arrowsmith, Cheryl H; Schmees, Norbert; Petersen, Kirstin.
Affiliation
  • Göricke F; Research & Development, Pharmaceuticals, Bayer AG, 42096 Wuppertal, Germany.
  • Vu V; Structural Genomics Consortium, University of Toronto, Toronto, Ontario M5G 1L7, Canada.
  • Smith L; Structural Genomics Consortium, University of Toronto, Toronto, Ontario M5G 1L7, Canada.
  • Scheib U; Nuvisan Innovation Campus Berlin, 13353 Berlin, Germany.
  • Böhm R; Nuvisan Innovation Campus Berlin, 13353 Berlin, Germany.
  • Akkilic N; Nuvisan Innovation Campus Berlin, 13353 Berlin, Germany.
  • Wohlfahrt G; Research & Development, Pharmaceuticals, Bayer AG, 13353 Berlin, Germany.
  • Weiske J; Nuvisan Innovation Campus Berlin, 13353 Berlin, Germany.
  • Bömer U; Nuvisan Innovation Campus Berlin, 13353 Berlin, Germany.
  • Brzezinka K; Nuvisan Innovation Campus Berlin, 13353 Berlin, Germany.
  • Lindner N; Research & Development, Pharmaceuticals, Bayer AG, 42096 Wuppertal, Germany.
  • Lienau P; Research & Development, Pharmaceuticals, Bayer AG, 13353 Berlin, Germany.
  • Gradl S; Research & Development, Pharmaceuticals, Bayer AG, 13353 Berlin, Germany.
  • Beck H; Research & Development, Pharmaceuticals, Bayer AG, 42096 Wuppertal, Germany.
  • Brown PJ; Structural Genomics Consortium, University of Toronto, Toronto, Ontario M5G 1L7, Canada.
  • Santhakumar V; Structural Genomics Consortium, University of Toronto, Toronto, Ontario M5G 1L7, Canada.
  • Vedadi M; Structural Genomics Consortium, University of Toronto, Toronto, Ontario M5G 1L7, Canada.
  • Barsyte-Lovejoy D; Department of Pharmacology and Toxicology, University of Toronto, Toronto, Ontario M5S 1A8, Canada.
  • Arrowsmith CH; Structural Genomics Consortium, University of Toronto, Toronto, Ontario M5G 1L7, Canada.
  • Schmees N; Structural Genomics Consortium, University of Toronto, Toronto, Ontario M5G 1L7, Canada.
  • Petersen K; Nuvisan Innovation Campus Berlin, 13353 Berlin, Germany.
J Med Chem ; 66(5): 3431-3447, 2023 03 09.
Article in En | MEDLINE | ID: mdl-36802665

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Signal Transduction / Ubiquitin-Specific Proteases Language: En Journal: J Med Chem Journal subject: QUIMICA Year: 2023 Document type: Article Affiliation country: Alemania Country of publication: Estados Unidos

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Signal Transduction / Ubiquitin-Specific Proteases Language: En Journal: J Med Chem Journal subject: QUIMICA Year: 2023 Document type: Article Affiliation country: Alemania Country of publication: Estados Unidos