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7-N-Substituted-3-oxadiazole Quinolones with Potent Antimalarial Activity Target the Cytochrome bc1 Complex.
Nguyen, William; Dans, Madeline G; Currie, Iain; Awalt, Jon Kyle; Bailey, Brodie L; Lumb, Chris; Ngo, Anna; Favuzza, Paola; Palandri, Josephine; Ramesh, Saishyam; Penington, Jocelyn; Jarman, Kate E; Mukherjee, Partha; Chakraborty, Arnish; Maier, Alexander G; van Dooren, Giel G; Papenfuss, Tony; Wittlin, Sergio; Churchyard, Alisje; Baum, Jake; Winzeler, Elizabeth A; Baud, Delphine; Brand, Stephen; Jackson, Paul F; Cowman, Alan F; Sleebs, Brad E.
Affiliation
  • Nguyen W; The Walter and Eliza Hall Institute of Medical Research, Parkville 3052, Australia.
  • Dans MG; Department of Medical Biology, The University of Melbourne, Parkville 3010, Australia.
  • Currie I; The Walter and Eliza Hall Institute of Medical Research, Parkville 3052, Australia.
  • Awalt JK; Department of Medical Biology, The University of Melbourne, Parkville 3010, Australia.
  • Bailey BL; The Walter and Eliza Hall Institute of Medical Research, Parkville 3052, Australia.
  • Lumb C; Department of Medical Biology, The University of Melbourne, Parkville 3010, Australia.
  • Ngo A; The Walter and Eliza Hall Institute of Medical Research, Parkville 3052, Australia.
  • Favuzza P; Department of Medical Biology, The University of Melbourne, Parkville 3010, Australia.
  • Palandri J; The Walter and Eliza Hall Institute of Medical Research, Parkville 3052, Australia.
  • Ramesh S; Department of Medical Biology, The University of Melbourne, Parkville 3010, Australia.
  • Penington J; The Walter and Eliza Hall Institute of Medical Research, Parkville 3052, Australia.
  • Jarman KE; The Walter and Eliza Hall Institute of Medical Research, Parkville 3052, Australia.
  • Mukherjee P; The Walter and Eliza Hall Institute of Medical Research, Parkville 3052, Australia.
  • Chakraborty A; Department of Medical Biology, The University of Melbourne, Parkville 3010, Australia.
  • Maier AG; The Walter and Eliza Hall Institute of Medical Research, Parkville 3052, Australia.
  • van Dooren GG; Department of Medical Biology, The University of Melbourne, Parkville 3010, Australia.
  • Papenfuss T; Research School of Biology, The Australian National University, Canberra 2600, Australia.
  • Wittlin S; The Walter and Eliza Hall Institute of Medical Research, Parkville 3052, Australia.
  • Churchyard A; Department of Medical Biology, The University of Melbourne, Parkville 3010, Australia.
  • Baum J; The Walter and Eliza Hall Institute of Medical Research, Parkville 3052, Australia.
  • Winzeler EA; Department of Medical Biology, The University of Melbourne, Parkville 3010, Australia.
  • Baud D; TCG Lifesciences, Kolkata, West Bengal 700091, India.
  • Brand S; TCG Lifesciences, Kolkata, West Bengal 700091, India.
  • Jackson PF; Research School of Biology, The Australian National University, Canberra 2600, Australia.
  • Cowman AF; Research School of Biology, The Australian National University, Canberra 2600, Australia.
  • Sleebs BE; The Walter and Eliza Hall Institute of Medical Research, Parkville 3052, Australia.
ACS Infect Dis ; 9(3): 668-691, 2023 03 10.
Article in En | MEDLINE | ID: mdl-36853190

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Malaria, Falciparum / Quinolones / Folic Acid Antagonists / Antimalarials Limits: Animals Language: En Journal: ACS Infect Dis Year: 2023 Document type: Article Affiliation country: Australia Country of publication: Estados Unidos

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Malaria, Falciparum / Quinolones / Folic Acid Antagonists / Antimalarials Limits: Animals Language: En Journal: ACS Infect Dis Year: 2023 Document type: Article Affiliation country: Australia Country of publication: Estados Unidos