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Subnanomolar Cathepsin S Inhibitors with High Selectivity: Optimizing Covalent Reversible α-Fluorovinylsulfones and α-Sulfonates as Potential Immunomodulators in Cancer.
Fuchs, Natalie; Meta, Mergim; Lantzberg, Bellinda; Bros, Matthias; Ling Kuan, Seah; Weil, Tanja; Schirmeister, Tanja.
Affiliation
  • Fuchs N; Institute of Pharmaceutical and Biomedical Sciences (IPBS), Johannes Gutenberg University Mainz, Staudingerweg 5, 55128, Mainz, Germany.
  • Meta M; Institute of Pharmaceutical and Biomedical Sciences (IPBS), Johannes Gutenberg University Mainz, Staudingerweg 5, 55128, Mainz, Germany.
  • Lantzberg B; Max Planck Institute for Polymer Research, Ackermannweg 10, 55128, Mainz, Germany.
  • Bros M; Department of Dermatology, University Medical Center Mainz, Langenbeckstr. 1, 55131, Mainz, Germany.
  • Ling Kuan S; Max Planck Institute for Polymer Research, Ackermannweg 10, 55128, Mainz, Germany.
  • Weil T; Max Planck Institute for Polymer Research, Ackermannweg 10, 55128, Mainz, Germany.
  • Schirmeister T; Institute of Pharmaceutical and Biomedical Sciences (IPBS), Johannes Gutenberg University Mainz, Staudingerweg 5, 55128, Mainz, Germany.
ChemMedChem ; 18(15): e202300160, 2023 08 01.
Article in En | MEDLINE | ID: mdl-37222230

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Cathepsins / Neoplasms Limits: Humans Language: En Journal: ChemMedChem Journal subject: FARMACOLOGIA / QUIMICA Year: 2023 Document type: Article Affiliation country: Alemania Country of publication: Alemania

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Cathepsins / Neoplasms Limits: Humans Language: En Journal: ChemMedChem Journal subject: FARMACOLOGIA / QUIMICA Year: 2023 Document type: Article Affiliation country: Alemania Country of publication: Alemania