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Development of an Affinity-Based Probe to Profile Endogenous Human Adenosine A3 Receptor Expression.
Beerkens, Bert L H; Snijders, Inge M; Snoeck, Joep; Liu, Rongfang; Tool, Anton T J; Le Dévédec, Sylvia E; Jespers, Willem; Kuijpers, Taco W; van Westen, Gerard J P; Heitman, Laura H; IJzerman, Adriaan P; van der Es, Daan.
Affiliation
  • Beerkens BLH; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, Einsteinweg 55, 2333 CC Leiden, The Netherlands.
  • Snijders IM; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, Einsteinweg 55, 2333 CC Leiden, The Netherlands.
  • Snoeck J; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, Einsteinweg 55, 2333 CC Leiden, The Netherlands.
  • Liu R; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, Einsteinweg 55, 2333 CC Leiden, The Netherlands.
  • Tool ATJ; Department of Molecular Hematology, Sanquin Research, Plesmalaan 125, 1066 CX Amsterdam, The Netherlands.
  • Le Dévédec SE; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, Einsteinweg 55, 2333 CC Leiden, The Netherlands.
  • Jespers W; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, Einsteinweg 55, 2333 CC Leiden, The Netherlands.
  • Kuijpers TW; Department of Molecular Hematology, Sanquin Research, Plesmalaan 125, 1066 CX Amsterdam, The Netherlands.
  • van Westen GJP; Department of Pediatric Immunology, Rheumatology and Infectious Diseases, Emma Children's Hospital, Academic Medical Center, University of Amsterdam, Amsterdam, The Netherlands, Meibergdreef 9, 1105 AZ Amsterdam, The Netherlands.
  • Heitman LH; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, Einsteinweg 55, 2333 CC Leiden, The Netherlands.
  • IJzerman AP; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, Einsteinweg 55, 2333 CC Leiden, The Netherlands.
  • van der Es D; Oncode Institute, Einsteinweg 55, 2333 CC Leiden, The Netherlands.
J Med Chem ; 66(16): 11399-11413, 2023 08 24.
Article in En | MEDLINE | ID: mdl-37531576

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Adenosine / Receptor, Adenosine A3 Limits: Humans Language: En Journal: J Med Chem Journal subject: QUIMICA Year: 2023 Document type: Article Affiliation country: Países Bajos

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Adenosine / Receptor, Adenosine A3 Limits: Humans Language: En Journal: J Med Chem Journal subject: QUIMICA Year: 2023 Document type: Article Affiliation country: Países Bajos