The reversible inhibitor SR-4835 binds Cdk12/cyclin K in a noncanonical G-loop conformation.
J Biol Chem
; 300(1): 105501, 2024 Jan.
Article
in En
| MEDLINE
| ID: mdl-38016516
Key words
Cdk10; Cdk12; Cdk13; DYRK1A; HIPK3; NVP-2; SR-4835; THZ1; THZ531; abemaciclib; cyclin K; dinaciclib; ribociclib; trilaciclib
Full text:
1
Collection:
01-internacional
Database:
MEDLINE
Main subject:
Cyclins
/
Cyclin-Dependent Kinases
/
Polyadenylation
Limits:
Humans
Language:
En
Journal:
J Biol Chem
Year:
2024
Document type:
Article
Affiliation country:
Alemania
Country of publication:
Estados Unidos